Abstract
Bleomycins are small glycopeptide cancer chemotherapeutics that give rise to 3'-modified DNA double-strand breaks (DSBs). In Saccharomyces cerevisiae, DSBs are predominantly repaired by RAD52-dependent homologous recombination (HR) with some support by Yku70/Yku80 (KU)-dependent pathways. The main DSB repair function of KU is believed to be as part of the non-homologous end-joining (NHEJ) pathway, but KU also functions in a "chromosome healing" pathway that seals DSBs by de novo telomere addition. We report here that rad52Deltayku70Delta double mutants are considerably more bleomycin hypersensitive than rad52Deltalig4Delta cells that lack the NHEJ-specific DNA ligase 4. Moreover, the telomere-specific KU mutation yku80-135i also dramatically increases rad52Delta bleomycin hypersensitivity, almost to the level of rad52Deltayku80Delta. The results indicate that telomere-specific functions of KU play a more prominent role in the repair of bleomycin-induced damage than its NHEJ functions, which could have important clinical implications for bleomycin-based combination chemotherapies.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Antibiotics, Antineoplastic / toxicity
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Antigens, Nuclear / genetics
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Antigens, Nuclear / physiology*
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Bleomycin / toxicity*
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DNA Damage*
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DNA Ligase ATP
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DNA Ligases / genetics
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DNA Ligases / physiology
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DNA Repair / genetics
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DNA Repair / physiology*
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DNA, Fungal / drug effects
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DNA, Fungal / genetics
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DNA, Fungal / metabolism
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DNA-Binding Proteins / genetics
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DNA-Binding Proteins / physiology*
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Ku Autoantigen
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Microbial Viability / drug effects
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Microbial Viability / genetics
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Mutation
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Rad52 DNA Repair and Recombination Protein / genetics
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Rad52 DNA Repair and Recombination Protein / physiology
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Recombination, Genetic
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Saccharomyces cerevisiae / drug effects
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Saccharomyces cerevisiae / genetics
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Saccharomyces cerevisiae / growth & development
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Saccharomyces cerevisiae Proteins / genetics
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Saccharomyces cerevisiae Proteins / physiology
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Telomere / genetics
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Telomere / metabolism*
Substances
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Antibiotics, Antineoplastic
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Antigens, Nuclear
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DNA, Fungal
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DNA-Binding Proteins
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RAD52 protein, S cerevisiae
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Rad52 DNA Repair and Recombination Protein
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Saccharomyces cerevisiae Proteins
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Bleomycin
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Ku Autoantigen
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DNA Ligases
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DNA Ligase ATP