3-Nitropropionic acid activates calpain/cdk5 pathway in rat striatum

Neurosci Lett. 2007 Jun 21;421(1):77-81. doi: 10.1016/j.neulet.2007.05.038. Epub 2007 May 26.

Abstract

3-Nitropropionic acid (3-NP) is a neurotoxin that inhibits mitochondrial complex II and is used in an experimental model of Huntington's disease. Treatment of rats with 3-NP 30mgkg(-1) i.p. once a day for 5 days induced an increase in calpain activation in rat striatum, measured by the formation of 145kDa fragment of alpha-spectrin breakdown and by an increase in enzymatic calpain activity. In this neurotoxic model, Western blot studies revealed that calpain activity increase was followed by changes in cyclin-dependent kinase 5 (cdk5) and its activator p25. Our results indicated, after 10 days of treatment with 3-NP, a decrease in myocyte enhancer factor phosphorylation, a neuronal prosurvival factor. Thus, a decrease in its expression indicates a new potential mechanism of neuronal cell death mediated by the neurotoxin 3-NP. Accordingly, in our study we demonstrated in rat striatum the activation of the calpain/cdk5/p25 pathway in the 3-NP model. Previous studies have linked the deregulation of cdk5 with neurodegenerative diseases, such as Alzheimer's and Parkinson's. We suggest that calpain/cdk5 activation could also be a common pathway activated in other neurodegenerative diseases, which is liable to be targeted.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analysis of Variance
  • Animals
  • Calpain / metabolism*
  • Convulsants / pharmacology*
  • Corpus Striatum / drug effects*
  • Cyclin-Dependent Kinase 5 / metabolism*
  • Enzyme Activation / drug effects
  • Male
  • Nitro Compounds / pharmacology*
  • Propionates / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Signal Transduction / drug effects*
  • Time Factors

Substances

  • Convulsants
  • Nitro Compounds
  • Propionates
  • Cyclin-Dependent Kinase 5
  • Calpain
  • 3-nitropropionic acid