Variability in secondary structure of the antimicrobial peptide Cateslytin in powder, solution, DPC micelles and at the air-water interface

Eur Biophys J. 2007 Nov;36(8):1019-27. doi: 10.1007/s00249-007-0169-8. Epub 2007 Jul 7.

Abstract

Cateslytin (bCGA (344)RSMRLSFRARGYGFR(358)), a five positively charged 15 amino-acid residues arginine-rich antimicrobial peptide, was synthesized using a very efficient procedure leading to high yields and to a 99% purity as determined by HPLC and mass spectrometry. Circular dichroism, polarized attenuated total reflectance fourier transformed infrared, polarization modulation infrared reflection Absorption spectroscopies and proton two-dimensional NMR revealed the flexibility of such a peptide. Whereas being mostly disordered as a dry powder or in water solution, the peptide acquires a alpha-helical character in the "membrane mimicking" solvent trifuoroethanol. In zwitterionic micelles of dodecylphophatidylcholine the helical character is retained but to a lesser extent, the peptide returning mainly to its disordered state. A beta-sheet contribution of almost 100% is detected at the air-water interface. Such conformational plasticity is discussed regarding the antimicrobial action of Cateslytin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Air
  • Amino Acid Sequence
  • Anti-Bacterial Agents / chemical synthesis
  • Anti-Bacterial Agents / chemistry*
  • Chromogranin A / chemical synthesis
  • Chromogranin A / chemistry*
  • Circular Dichroism
  • Magnetic Resonance Spectroscopy
  • Micelles
  • Molecular Sequence Data
  • Peptide Fragments / chemical synthesis
  • Peptide Fragments / chemistry*
  • Pharmaceutical Solutions
  • Powders
  • Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
  • Spectrophotometry, Atomic
  • Spectroscopy, Fourier Transform Infrared
  • Trifluoroethanol / chemistry
  • Water

Substances

  • Anti-Bacterial Agents
  • Chromogranin A
  • Micelles
  • Peptide Fragments
  • Pharmaceutical Solutions
  • Powders
  • chromogranin A (344-358)
  • Water
  • Trifluoroethanol