Multi-drug resistance mediated by P-glycoprotein overexpression is not correlated with ZAP-70/CD38 expression in B-cell chronic lymphocytic leukemia

Leuk Lymphoma. 2007 Aug;48(8):1556-60. doi: 10.1080/10428190701457931.

Abstract

ZAP-70 and CD38 expression can identify B-cell chronic lymphocytic leukemia with an inferior clinical outcome. Many groups have investigated the meaning of the expression of these two proteins and the correlation with the bad prognosis in B-CLL. But nobody has investigated the relation between the multidrug resistance mediated by Pgp overexpression (MDR1) and ZAP-70/CD38 coexpression. Forty-one untreated and stage A patients, either ZAP-70(+)CD38(+) or ZAP-70(-)CD38(-), were tested to determine the MDR1 status. MDR1 was observed in 41% of CLL ZAP-70(+)CD38(+) and in 37% of CLL ZAP-70(-)CD38(-). The difference was not significant (p = 0.745). Patients with ZAP-70 and CD38 positive CLL can not be candidates for MDR1 antagonists.

MeSH terms

  • ADP-ribosyl Cyclase 1 / metabolism*
  • ATP Binding Cassette Transporter, Subfamily B
  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / metabolism*
  • Aged
  • Aged, 80 and over
  • Drug Resistance, Multiple*
  • Drug Resistance, Neoplasm
  • Female
  • Gene Expression Regulation, Leukemic*
  • Humans
  • Immunoblotting
  • Leukemia, Lymphocytic, Chronic, B-Cell / metabolism*
  • Male
  • Membrane Glycoproteins / metabolism*
  • Middle Aged
  • Prognosis
  • Up-Regulation
  • ZAP-70 Protein-Tyrosine Kinase / metabolism*

Substances

  • ABCB1 protein, human
  • ATP Binding Cassette Transporter, Subfamily B
  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • Membrane Glycoproteins
  • ZAP-70 Protein-Tyrosine Kinase
  • ZAP70 protein, human
  • CD38 protein, human
  • ADP-ribosyl Cyclase 1