HIF-dependent antitumorigenic effect of antioxidants in vivo

Cancer Cell. 2007 Sep;12(3):230-8. doi: 10.1016/j.ccr.2007.08.004.

Abstract

The antitumorigenic activity of antioxidants has been presumed to arise from their ability to squelch DNA damage and genomic instability mediated by reactive oxygen species (ROS). Here, we report that antioxidants inhibited three tumorigenic models in vivo. Inhibition of a MYC-dependent human B lymphoma model was unassociated with genomic instability but was linked to diminished hypoxia-inducible factor (HIF)-1 levels in a prolyl hydroxylase 2 and von Hippel-Lindau protein-dependent manner. Ectopic expression of an oxygen-independent, stabilized HIF-1 mutant rescued lymphoma xenografts from inhibition by two antioxidants: N-acetylcysteine and vitamin C. These findings challenge the paradigm that antioxidants diminish tumorigenesis primarily through decreasing DNA damage and mutations and provide significant support for a key antitumorigenic effect of diminishing HIF levels.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Acetylcysteine / pharmacology*
  • Animals
  • Antineoplastic Agents / pharmacology*
  • Antioxidants / pharmacology*
  • Ascorbic Acid / pharmacology*
  • Cell Line
  • Genomic Instability
  • Humans
  • Hypoxia-Inducible Factor 1 / genetics
  • Hypoxia-Inducible Factor 1 / metabolism
  • Hypoxia-Inducible Factor 1 / physiology*
  • Mice
  • Mice, Transgenic
  • Mutation

Substances

  • Antineoplastic Agents
  • Antioxidants
  • Hypoxia-Inducible Factor 1
  • Ascorbic Acid
  • Acetylcysteine

Associated data

  • GEO/GSE8627