A Polypodium leucotomos extract inhibits solar-simulated radiation-induced TNF-alpha and iNOS expression, transcriptional activation and apoptosis

Exp Dermatol. 2007 Oct;16(10):823-9. doi: 10.1111/j.1600-0625.2007.00603.x.

Abstract

In this report, we have examined the molecular basis of the photoprotective effect of a hydrophilic extract of the fern Polypodium leucotomos (PL) in vitro, using a solar simulator as the source of UV radiation (SSR). We found that pretreatment of human keratinocytes with PL inhibited SSR-mediated increase of tumor necrosis factor (TNF)-alpha and also abrogated nitric oxide (NO) production. Consistent with this, PL blocked the induction of inducible nitric oxide synthase (iNOS) elicited by SSR. In addition, PL inhibited the SSR-mediated transcriptional activation of NF-kappaB and AP1. Finally, we demonstrated that pretreatment with PL exerted a cytoprotective effect against SSR-induced damage, resulting in increased cell survival. Together, these data postulate a multifactor mechanism of protection not exclusively reliant on the antioxidant capability of PL, and strengthen the basic knowledge on the photoprotective effect of this botanical agent.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / drug effects*
  • Apoptosis / radiation effects
  • Ascorbic Acid / pharmacology
  • Cell Line
  • Cell Survival / drug effects
  • Cell Survival / radiation effects
  • Dose-Response Relationship, Drug
  • Gene Expression / drug effects
  • Gene Expression / radiation effects
  • Humans
  • Keratinocytes / drug effects*
  • Keratinocytes / metabolism
  • Keratinocytes / radiation effects
  • Luciferases / genetics
  • Luciferases / metabolism
  • NF-kappa B / genetics
  • NF-kappa B / metabolism
  • Nitric Oxide / metabolism
  • Nitric Oxide Synthase Type II / metabolism*
  • Plant Extracts / pharmacology*
  • Plant Leaves / chemistry
  • Polypodium / chemistry*
  • Sunlight
  • Transcription Factor AP-1 / genetics
  • Transcription Factor AP-1 / metabolism
  • Transcription, Genetic / drug effects
  • Transcription, Genetic / radiation effects
  • Tumor Necrosis Factor-alpha / metabolism*
  • Ultraviolet Rays

Substances

  • NF-kappa B
  • Plant Extracts
  • Transcription Factor AP-1
  • Tumor Necrosis Factor-alpha
  • Nitric Oxide
  • Luciferases
  • Nitric Oxide Synthase Type II
  • Ascorbic Acid