[Clozapine and selective serotonin reuptake inhibitors: risks of toxicity]

Tijdschr Psychiatr. 2007;49(9):655-9.
[Article in Dutch]

Abstract

A 25-year-old woman, known to have schizoaffective disorder, presented with symptoms that had arisen a few weeks earlier. The symptoms indicated that she had a toxic clozapine blood level. The probable cause of the toxicity was a pharmacokinetic interaction between citalopram and clozapine at the level of the cytochrome P450 system. A literature search reveals the importance of monitoring the interactions between selective serotonin reuptake inhibitors and clozapine, a procedure which should, if possible, be accompanied by blood level measurements. Caution is called for, particularly when non-smokers are involved.

Publication types

  • Case Reports
  • English Abstract

MeSH terms

  • Adult
  • Antipsychotic Agents / adverse effects
  • Antipsychotic Agents / blood
  • Antipsychotic Agents / pharmacokinetics
  • Clozapine / adverse effects
  • Clozapine / blood
  • Clozapine / pharmacokinetics*
  • Cytochrome P-450 Enzyme Inhibitors*
  • Drug Interactions
  • Enzyme Inhibitors / adverse effects
  • Enzyme Inhibitors / blood
  • Enzyme Inhibitors / pharmacokinetics*
  • Female
  • Humans
  • Psychotic Disorders / drug therapy*
  • Selective Serotonin Reuptake Inhibitors / adverse effects
  • Selective Serotonin Reuptake Inhibitors / blood
  • Selective Serotonin Reuptake Inhibitors / pharmacokinetics*

Substances

  • Antipsychotic Agents
  • Cytochrome P-450 Enzyme Inhibitors
  • Enzyme Inhibitors
  • Serotonin Uptake Inhibitors
  • Clozapine