Assessment of radionuclidic impurities in 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG) routine production

Appl Radiat Isot. 2008 Mar;66(3):295-302. doi: 10.1016/j.apradiso.2007.08.015. Epub 2007 Sep 4.

Abstract

In this paper, radionuclidic impurities generated during the bombardment of [18 O]water in the routine production of 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG) were studied. In order to assess such impurities and the efficacy of purification methods through the different steps of the synthesis, samples of the target filters, purification columns, [18 O]water recovered after the synthesis, and the final solution was collected and their activities measured and analyzed by means of a gamma-ray spectrometry system. The data demonstrated that purification methods adopted for the synthesis provide the [18F]FDG radionuclidically pure, as requested by the EU Pharmacopeia.

MeSH terms

  • Fluorodeoxyglucose F18 / chemical synthesis*
  • Fluorodeoxyglucose F18 / isolation & purification
  • Oxygen / chemistry
  • Radiopharmaceuticals / chemical synthesis*
  • Radiopharmaceuticals / isolation & purification
  • Spectrometry, Gamma

Substances

  • Radiopharmaceuticals
  • Fluorodeoxyglucose F18
  • Oxygen