Activation of the p53 pathway down-regulates the osteoprotegerin expression and release by vascular endothelial cells

Blood. 2008 Feb 1;111(3):1287-94. doi: 10.1182/blood-2007-05-092031. Epub 2007 Nov 13.

Abstract

It has been shown that the expression of osteoprotegerin (OPG) is up-regulated in tumor-associated endothelial cells as well as in the sera of patients affected by both solid tumors and hematologic malignancies. We now report that sera of p53(-/-) mice contain higher levels of OPG with respect to p53(+/+) mice and that endothelial cells, in which p53 was knocked down by siRNA, release increased levels of OPG with respect to mock-transfected cells. Conversely, activation of the p53 pathway by the MDM2 small molecule antagonist Nutlin-3 significantly attenuated both spontaneous and tumor necrosis factor-alpha (TNF-alpha)-induced OPG mRNA and protein release in endothelial cell cultures. OPG promoter functional assays and chromatin immunoprecipitation experiments revealed inhibitory effects of Nutlin-3 on the TNF-alpha-induced NF-kappaB DNA binding activity to the OPG promoter. Because OPG inhibits the pro-tumoricidal activity of TNF-related apoptosis-inducing ligand, our findings suggest that, besides its well-documented functions within the malignant cancer cells, the ability of p53 to down-modulate OPG production by endothelial cells may be an additional important mechanism whereby it exerts non-cell-autonomous tumor suppression function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Cycle
  • Cells, Cultured
  • Cytokines / metabolism
  • Down-Regulation* / drug effects
  • Endothelial Cells / cytology
  • Endothelial Cells / metabolism*
  • Humans
  • Imidazoles / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • NF-kappa B / metabolism
  • Osteoprotegerin / metabolism*
  • Piperazines / metabolism
  • Promoter Regions, Genetic / genetics
  • Signal Transduction* / drug effects
  • Tumor Necrosis Factor-alpha / pharmacology
  • Tumor Suppressor Protein p53 / deficiency
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • Cytokines
  • Imidazoles
  • NF-kappa B
  • Osteoprotegerin
  • Piperazines
  • Tumor Necrosis Factor-alpha
  • Tumor Suppressor Protein p53
  • nutlin 3