The characterization of crude products from solid-phase peptide synthesis by mu-HPLC/fast atom bombardment mass spectrometry

Pept Res. 1991 Jan-Feb;4(1):40-6.

Abstract

Crude product mixtures from the solid-phase synthesis of a series of peptides were analyzed by on-line packed, fused silica column mu-HPLC/Continuous Flow Fast Atom Bombardment Mass Spectrometry (mu-HPLC/CF-FABMS). The technique is superior to the direct FAB analysis of crude product mixtures since competitive ionization and suppression effects are not generally observed. Positive correlation between a chromatographic peak and the desired synthetic product may be obtained. An accurate assessment of peptide deprotection can be made without ambiguity arising from the MS fragmentation of the more labile t-butyl and BOC protecting groups used in FMOC-based solid-phase peptide synthesis strategies. mu-HPLC combined with in-line UV detection and MS analysis allows the use of minimum sample and injection volumes, typically 10-50 pmol contained in 0.2-0.5 microliters.

MeSH terms

  • Amino Acid Sequence
  • Chromatography, High Pressure Liquid / methods*
  • Molecular Sequence Data
  • Oligopeptides / analysis*
  • Oligopeptides / chemical synthesis
  • Oligopeptides / chemistry
  • Peptides, Cyclic / analysis
  • Peptides, Cyclic / chemical synthesis
  • Peptides, Cyclic / chemistry
  • Spectrometry, Mass, Fast Atom Bombardment / methods*

Substances

  • Oligopeptides
  • Peptides, Cyclic