Conjugated polyelectrolyte based real-time fluorescence assay for phospholipase C

Anal Chem. 2008 Jan 1;80(1):150-8. doi: 10.1021/ac701672g. Epub 2007 Nov 29.

Abstract

A fluorescence turnoff assay for phospholipase C (PLC) from Clostridium perfringens is developed based on the reversible interaction between the natural substrate, phosphatidylcholine, and a fluorescent, water-soluble conjugated polyelectrolyte (CPE). The fluorescence intensity of the CPE in water is increased substantially by the addition of the phospholipid due to the formation of a CPE-lipid complex. Incubation of the CPE-lipid complex with the enzyme PLC causes the fluorescence intensity to decrease (turnoff sensor); the response arises due to PLC-catalyzed hydrolysis of the phosphatidylcholine, which effectively disrupts the CPE-lipid complex. The PLC assay operates with phospholipid substrate concentrations in the micromolar range, and the analytical detection limit for PLC is <1 nM. The optimized assay provides a convenient, rapid, and real-time sensor for PLC activity. The real-time fluorescence intensity from the CPE can be converted to substrate concentration by using an ex situ calibration curve, allowing PLC-catalyzed reaction rates and kinetic parameters to be determined. PLC activation by Ca2+ and inhibition by EDTA and fluoride ion are demonstrated using the optimized sensor.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Anions / chemistry
  • Catalysis
  • Cattle
  • Clostridium perfringens / enzymology
  • Electrolytes / chemical synthesis
  • Electrolytes / chemistry*
  • Fluorescence
  • Hydrolysis
  • Kinetics
  • Phospholipid Ethers / chemistry
  • Phospholipid Ethers / metabolism
  • Polymers / chemical synthesis
  • Polymers / chemistry*
  • Solubility
  • Solutions
  • Type C Phospholipases / analysis
  • Type C Phospholipases / antagonists & inhibitors
  • Type C Phospholipases / chemistry*
  • Type C Phospholipases / metabolism*
  • Water / chemistry

Substances

  • 1,2-dihexadecyl-sn-glycero-3-phosphocholine
  • Anions
  • Electrolytes
  • Phospholipid Ethers
  • Polymers
  • Solutions
  • Water
  • Type C Phospholipases