Suppression of plasma matrix metalloproteinase-9 following montelukast treatment in childhood asthma

Pediatr Int. 2007 Dec;49(6):918-22. doi: 10.1111/j.1442-200X.2007.02497.x.

Abstract

Background: Montelukast and ketotifen are commonly prescribed anti-inflammatory medications used in the treatment of childhood asthma.

Methods: To investigate the modulation effect of montelukast and ketotifen, the levels of exhaled nitric oxide (eNO) and plasma matrix metalloproteinase-9 (MMP-9) were analyzed in a group of 30 children with mild persistent asthma.

Results: Patients on montelukast therapy for 8 weeks had significantly decreased levels of eNO and plasma MMP-9, which were associated with improved symptoms and enhanced peak expiratory flow but not significantly associated with increased level of tissue inhibitor metalloproteinase-1 (TIMP-1). In contrast, treatment with ketotifen produced no significant changes in these parameters until 4-6 weeks into the therapy and no effect on plasma MMP-9.

Conclusion: Leukotriene antagonists, such as montelukast, may be better non-steroidal anti-inflammatory drugs for preventing airway inflammation in mild childhood asthma.

MeSH terms

  • Acetates / pharmacology*
  • Acetates / therapeutic use
  • Adolescent
  • Anti-Asthmatic Agents / pharmacology*
  • Anti-Asthmatic Agents / therapeutic use
  • Asthma / drug therapy*
  • Asthma / metabolism
  • Breath Tests
  • Child
  • Cyclopropanes
  • Female
  • Histamine H1 Antagonists / pharmacology
  • Histamine H1 Antagonists / therapeutic use
  • Humans
  • Ketotifen / pharmacology
  • Ketotifen / therapeutic use
  • Leukotriene Antagonists / pharmacology*
  • Leukotriene Antagonists / therapeutic use
  • Male
  • Matrix Metalloproteinase 9 / blood*
  • Nitric Oxide / analysis
  • Peak Expiratory Flow Rate
  • Quinolines / pharmacology*
  • Quinolines / therapeutic use
  • Severity of Illness Index
  • Statistics, Nonparametric
  • Sulfides
  • Tissue Inhibitor of Metalloproteinase-1 / blood

Substances

  • Acetates
  • Anti-Asthmatic Agents
  • Cyclopropanes
  • Histamine H1 Antagonists
  • Leukotriene Antagonists
  • Quinolines
  • Sulfides
  • Tissue Inhibitor of Metalloproteinase-1
  • Nitric Oxide
  • Matrix Metalloproteinase 9
  • montelukast
  • Ketotifen