Magnesium and potassium ions on tone and reactivity of human placental chorionic veins

Gen Pharmacol. 1991;22(6):1121-5. doi: 10.1016/0306-3623(91)90588-w.

Abstract

1. In vitro studies were undertaken to investigate the effects of external potassium [K+]0 2.4-7.1 mM and magnesium [Mg2+]0 0-4.8 mM concentration on human chorionic veins basal tone and on serotonin (5-HT)-induced contractions. 2. The higher the [Mg2+]0, the less the basal tension developed in isolated chorionic veins, irrespective of the [K+]0. 3. The EC50 value to 5-HT was enhanced by increases in [Mg2+]0, whereas the ability of 5-HT to induce a maximal contraction was attenuated. 4. The rightward shift of the concentration-response curves and reduced Emax response, observed when the concentration of [Mg2+]0 was raised, indicate a non-competitive antagonism of [Mg2+]0 with 5-HT. 5. The lack of an effect of [K+]0 on the EC50 and Emax values for 5-HT suggest that in this tissue the affinity of 5-HT for 5-HT receptors does not involve potassium. 6. These results suggest that basal tone and 5-HT-induced contractions of human chorionic vascular smooth muscle cells appear to be highly sensitive to alterations in extracellular Mg2+.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Chorionic Villi / physiology
  • Female
  • Humans
  • In Vitro Techniques
  • Magnesium / pharmacology*
  • Muscle Contraction / drug effects
  • Muscle Tonus / drug effects
  • Muscle, Smooth, Vascular / drug effects*
  • Placenta / blood supply
  • Potassium / pharmacology*
  • Pregnancy
  • Serotonin / pharmacology
  • Veins / drug effects

Substances

  • Serotonin
  • Magnesium
  • Potassium