Dietary n-3 polyunsaturated fatty acids and direct renin inhibition improve electrical remodeling in a model of high human renin hypertension

Hypertension. 2008 Feb;51(2):540-6. doi: 10.1161/HYPERTENSIONAHA.107.103143. Epub 2007 Dec 24.

Abstract

We compared the effect n-3 polyunsaturated fatty acids (PUFAs) with direct renin inhibition on electrophysiological remodeling in angiotensin II-induced cardiac injury. We treated double-transgenic rats expressing the human renin and angiotensinogen genes (dTGRs) from week 4 to 7 with n-3 PUFA ethyl-esters (Omacor; 25-g/kg diet) or a direct renin inhibitor (aliskiren; 3 mg/kg per day). Sprague-Dawley rats were controls. We performed electrocardiographic, magnetocardiographic, and programmed electrical stimulation. Dietary n-3 PUFAs increased the cardiac content of eicosapentaenoic and docosahexaenoic acid. At week 7, mortality in dTGRs was 31%, whereas none of the n-3 PUFA- or aliskiren-treated dTGRs died. Systolic blood pressure was modestly reduced in n-3 PUFA-treated (180+/-3 mm Hg) compared with dTGRs (208+/-5 mm Hg). Aliskiren-treated dTGRs and Sprague-Dawley rats were normotensive (110+/-3 and 119+/-6 mm Hg, respectively). Both n-3 PUFA-treated and untreated dTGRs showed cardiac hypertrophy and increased atrial natriuretic peptide levels. Prolonged QRS and QT(c) intervals and increased T-wave dispersion in dTGRs were reduced by n-3 PUFAs or aliskiren. Both treatments reduced arrhythmia induction from 75% in dTGRs to 17% versus 0% in Sprague-Dawley rats. Macrophage infiltration and fibrosis were reduced by n-3 PUFAs and aliskiren. Connexin 43, a mediator of intermyocyte conduction, was redistributed to the lateral cell membranes in dTGRs. n-3 PUFAs and aliskiren restored normal localization to the intercalated disks. Thus, n-3 PUFAs and aliskiren improved electrical remodeling, arrhythmia induction, and connexin 43 expression, despite a 70-mm Hg difference in blood pressure and the development of cardiac hypertrophy.

MeSH terms

  • Amides / pharmacology
  • Angiotensinogen / genetics
  • Angiotensinogen / metabolism
  • Animals
  • Animals, Genetically Modified
  • Antihypertensive Agents / pharmacology
  • Arrhythmias, Cardiac / etiology
  • Blood Pressure / drug effects
  • Cardiac Pacing, Artificial
  • Cardiomegaly / etiology
  • Connexin 43 / metabolism
  • Dietary Fats / pharmacology*
  • Disease Models, Animal
  • Electrocardiography
  • Electrophysiology
  • Fatty Acids, Omega-3 / pharmacology*
  • Fumarates / pharmacology
  • Humans
  • Hypertension / complications
  • Hypertension / metabolism
  • Hypertension / mortality
  • Hypertension / physiopathology*
  • Magnetocardiography
  • Male
  • Rats
  • Rats, Sprague-Dawley
  • Renin / antagonists & inhibitors*
  • Renin / genetics
  • Renin / metabolism*
  • Up-Regulation

Substances

  • Amides
  • Antihypertensive Agents
  • Connexin 43
  • Dietary Fats
  • Fatty Acids, Omega-3
  • Fumarates
  • Angiotensinogen
  • aliskiren
  • Renin