Enantioselective behavioral effects of threo-methylphenidate in rats

Pharmacol Biochem Behav. 1991 Dec;40(4):875-80. doi: 10.1016/0091-3057(91)90100-g.

Abstract

The relative potency of d- and l-threo-methylphenidate (d-MPH and l-MPH) was evaluated using three behavioral paradigms for rats: Responding maintained by a fixed-interval schedule of reinforcement (FI), responding maintained by a concurrent variable-interval schedule of reinforcement (Conc VI VI), and consumption of sweetened condensed milk during a 15-min free-access period. In each case the potency of the d-MPH enantiomer greatly exceeded that of the l-MPH enantiomer. Temporal control of responding was reduced (FI) choice responding was equalized for most rats (Conc VI VI), and milk consumption was suppressed by d-MPH and dl-MPH.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Anorexia / chemically induced
  • Appetite / drug effects
  • Appetite Depressants / toxicity
  • Behavior, Animal / drug effects*
  • Male
  • Methylphenidate / chemistry
  • Methylphenidate / pharmacology*
  • Methylphenidate / toxicity
  • Rats
  • Reinforcement Schedule
  • Stereoisomerism

Substances

  • Appetite Depressants
  • Methylphenidate