Effects of PP-56 and vitamin E on platelet hyperaggregability, fatty acid abnormalities, and clinical manifestations in streptozocin-induced diabetic rats

Diabetes. 1991 Feb;40(2):233-9. doi: 10.2337/diab.40.2.233.

Abstract

The effects of vitamin E and D-myo-inositol 1,2,6-trisphosphate (PP-56) were investigated in long-term studies in streptozocin-induced diabetic rats fed a purified diet with 33% lipids and a polyunsaturated-to -saturated fatty acid ratio of 1. A supplement of vitamin E decreased plasma triglycerides, platelet lipid biosynthesis, some of the delta 6- and delta 5-desaturase abnormalities, and urine ketone bodies but did not affect the response of platelets to aggregation. PP-56 completely normalized the platelet reactivity to ADP and thrombin. This was accompanied by normalization of platelet lipid biosynthesis and diabetes-induced abnormalities in delta 6- and delta 5-desaturases. PP-56 treatment also reduced the mortality rate and to a certain extent urinary ketone bodies. The protective effect of PP-56 on platelet aggregation and mortality rate were dose related. PP-56, a molecule derived from phytic acid, seems to exert potent protective effects on some of the manifestations associated with diabetes in rats.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Diphosphate / pharmacology
  • Animals
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism
  • Calcium / metabolism
  • Diabetes Mellitus, Experimental / blood*
  • Diabetes Mellitus, Experimental / metabolism
  • Diabetes Mellitus, Experimental / pathology
  • Diet
  • Dose-Response Relationship, Drug
  • Fatty Acids / metabolism*
  • Inositol Phosphates / pharmacology
  • Lipids / blood
  • Male
  • Platelet Aggregation / drug effects*
  • Rats
  • Rats, Inbred Strains
  • Streptozocin
  • Thrombin / pharmacology
  • Vitamin E / pharmacology*

Substances

  • Fatty Acids
  • Inositol Phosphates
  • Lipids
  • Vitamin E
  • Streptozocin
  • Adenosine Diphosphate
  • Thrombin
  • Calcium
  • atrinositol