Potassium channel phosphorylation in excitable cells: providing dynamic functional variability to a diverse family of ion channels

Physiology (Bethesda). 2008 Feb:23:49-57. doi: 10.1152/physiol.00031.2007.

Abstract

Phosphorylation of potassium channels affects their function and plays a major role in regulating cell physiology. Here, we review previous studies of potassium channel phosphorylation, focusing first on studies employing site-directed mutagenesis of recombinant channels expressed in heterologous cells. We then discuss recent mass spectrometric-based approaches to identify and quantify phosphorylation at specific sites on native and recombinant potassium channels, and newly developed mass spectrometric-based techniques that may prove beneficial to future studies of potassium channel phosphorylation, its regulation, and its mechanism of channel modulation.

Publication types

  • Research Support, N.I.H., Extramural
  • Review

MeSH terms

  • Animals
  • Humans
  • Ion Channel Gating*
  • Mass Spectrometry / methods
  • Membrane Potentials
  • Models, Molecular
  • Mutation
  • Phosphorylation
  • Potassium Channels / chemistry
  • Potassium Channels / genetics
  • Potassium Channels / metabolism*
  • Protein Conformation
  • Protein Transport
  • Recombinant Proteins / metabolism
  • Time Factors

Substances

  • Potassium Channels
  • Recombinant Proteins