Comparison of the effects of ANF 99-126 and ANF 103-126 on captopril-induced renin release in man

Clin Endocrinol (Oxf). 1991 Jun;34(6):493-9. doi: 10.1111/j.1365-2265.1991.tb00330.x.

Abstract

Objective: The aim was to examine the effects of atrial natriuretic factor (ANF) 99-126 and ANF 103-126, an N-terminal shortened analogue of the peptide, on the plasma renin activity response to captopril, an inhibitor of angiotensin-converting enzyme.

Design: Two protocols were performed. In the first protocol, subjects were studied on three occasions. Captopril 25 mg was given and a 60 minute infusion of 5% D-glucose (placebo), or ANF 99-126 3 or 10 pmol/kg/min, was administered in a single blind randomized manner. The second protocol was divided in two parallel phases comparing ANF 103-126 either 3 or 10 pmol/kg/min to placebo.

Subjects: Thirty-three salt-replete healthy male volunteers aged 21-39 years were studied in the supine position.

Measurements: Plasma renin activity, plasma ANF 99-126 and ANF 103-126 levels, heart rate and blood pressure were measured.

Results: Compared to placebo infusion, the rise in plasma renin activity after captopril was attenuated by ANF 99-126 infusion (from 755% of baseline to 294% by ANF 99-126 3 pmol/kg/min and from 755 to 202% by 10 pmol/kg/min; P less than 0.03 and P less than 0.01 respectively). The comparable findings with ANF 103-126 were 492 to 218% (3 pmol/kg/min) and 645 to 364% (10 pmol/kg/min) (P less than 0.01 and P less than 0.01 respectively).

Conclusions: The results, taken in conjunction with previous findings, suggest that atrial natriuretic factor inhibits in a non-selective manner the renin response to all secretagogues so far tested in man. The current results also suggest that the anti-renin action of atrial natriuretic factor does not depend on the first four N-terminal amino acids of the native peptide.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Atrial Natriuretic Factor / pharmacology*
  • Blood Pressure / drug effects
  • Captopril / pharmacology*
  • Depression, Chemical
  • Diuretics / pharmacology*
  • Humans
  • Male
  • Peptide Fragments / pharmacology*
  • Renin / blood
  • Renin / metabolism*
  • Single-Blind Method
  • Supination

Substances

  • Diuretics
  • Peptide Fragments
  • atrial natriuretic factor prohormone (103-126)
  • Atrial Natriuretic Factor
  • Captopril
  • Renin