A novel tumor necrosis factor-alpha suppressant, ONO-SM362, prevents liver failure and promotes liver regeneration after extensive hepatectomy

Surgery. 2008 Apr;143(4):545-55. doi: 10.1016/j.surg.2007.11.010. Epub 2008 Feb 19.

Abstract

Background: Tumor necrosis factor (TNF)-alpha is a cytokine that initiates liver regeneration after hepatectomy (HTx), although extensive HTx can cause liver failure with significant rise in serum TNF-alpha levels. To test our hypothesis that modulation of endogenous TNF-alpha attenuates liver failure even after extensive HTx, we used ONO-SM362, a novel TNF-alpha inhibitor, in mice subjected to 85% HTx.

Methods: ICR mice were divided into 5 groups: 70% HTx, 85% HTx, 85% HTx plus ONO-SM362, 85% HTx plus monoclonal TNF-alpha antibody (mAb), and 85% HTx plus FR167653, a TNF-alpha inhibitor. We analyzed the survival rate, blood ammonia (NH(3)), serum TNF-alpha levels, TNF-alpha mRNA expression in the liver and spleen by real-time polymerase chain reaction, histologic changes, polymorphonuclear neutrophils (PMNs) infiltration, and proliferating cell nuclear antigen labeling index (PCNA LI) in the 5 groups.

Results: The survival rate at 7 days after surgery was 100%, 0%, 100%, 50%, and 0%, for the 70% HTx, 85% HTx, 85% HTx + ONO-SM362, 85% HTx + mAb, and 85% HTx + FR167653, respectively. Mice that underwent 85% HTx died from liver failure associated with a significant rise in serum TNF-alpha level. ONO-SM362 and mAb improved animal survival and enhanced PCNA LI. In addition, ONO-SM362 inhibited TNF-alpha mRNA expression in the remnant liver and suppressed PMNs infiltration.

Conclusions: Suppression of excessive TNF-alpha production using ONO-SM362 ameliorated liver failure after 85% HTx.

Publication types

  • Evaluation Study

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology*
  • Disease Models, Animal
  • Hepatectomy / adverse effects*
  • Liver Failure / etiology
  • Liver Failure / mortality
  • Liver Failure / prevention & control*
  • Liver Regeneration / drug effects*
  • Male
  • Mice
  • Mice, Inbred ICR
  • Organophosphorus Compounds / pharmacology
  • Organophosphorus Compounds / therapeutic use
  • Survival Analysis
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors*

Substances

  • (1S,2R)-2-hexyloxy carbonylamino-1 methyl-2-(3-methoxyphenyl) ethyl disodium phosphate
  • Anti-Inflammatory Agents
  • Organophosphorus Compounds
  • Tumor Necrosis Factor-alpha