Effects of conformational activation of integrin alpha 1I and alpha 2I domains on selective recognition of laminin and collagen subtypes

Exp Cell Res. 2008 May 1;314(8):1734-43. doi: 10.1016/j.yexcr.2008.01.025. Epub 2008 Feb 9.

Abstract

Collagen receptor integrins alpha 1 beta 1 and alpha 2 beta 1 can selectively recognize different collagen subtypes. Here we show that their alpha I domains can discriminate between laminin isoforms as well: alpha 1I and alpha 2I recognized laminin-111, -211 and -511, whereas their binding to laminin-411 was negligible. Residue Arg-218 in alpha1 was found to be instrumental in high-avidity binding. The gain-of-function mutation E318W makes the alpha 2I domain to adopt the "open" high-affinity conformation, while the wild-type alpha 2I domain favors the "closed" low-affinity conformation. The E318W mutation markedly increased alpha 2I domain binding to the laminins (-111, -211 and -511), leading us to propose that the activation state of the alpha 2 beta 1 integrin defines its role as a laminin receptor. However, neither wild-type nor alpha 2IE318W domain could bind to laminin-411. alpha 2IE318W also bound tighter to all collagens than alpha 2I wild-type, but it showed reduced ability to discriminate between collagens I, IV and IX. The corresponding mutation, E317A, in the alpha 1I domain transformed the domain into a high-avidity binder of collagens I and IV. Thus, our results indicate that conformational activation of integrin alpha 1I and alpha 2I domains leads to high-avidity binding to otherwise disfavored collagen subtypes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Arginine / chemistry
  • Collagen / classification
  • Collagen / metabolism*
  • Humans
  • Integrin alpha1 / chemistry*
  • Integrin alpha1 / genetics
  • Integrin alpha1 / metabolism
  • Integrin alpha2 / chemistry*
  • Integrin alpha2 / genetics
  • Integrin alpha2 / metabolism
  • Laminin / metabolism*
  • Models, Molecular
  • Mutation
  • Protein Binding
  • Protein Isoforms / metabolism
  • Protein Structure, Tertiary

Substances

  • Integrin alpha1
  • Integrin alpha2
  • Laminin
  • Protein Isoforms
  • laminin 1
  • laminin 10
  • laminin 8
  • Collagen
  • Arginine