The functional variant (Asp299gly) of toll-like receptor 4 (TLR4) influences TLR4-mediated cytokine production in rheumatoid arthritis

J Rheumatol. 2008 Apr;35(4):558-61. Epub 2008 Mar 15.

Abstract

Objective: To investigate functional consequences of the Toll-like receptor 4 (TLR4) variant (Asp299Gly) in rheumatoid arthritis (RA).

Methods: Peripheral blood mononuclear cells from 28 patients with RA carrying or not carrying the TLR4 variant were incubated with lipopolysaccharide (LPS) and heat shock protein B8 (HSPB8). Concentrations of interleukin 6 (IL-6), tumor necrosis factor-alpha(TNF-alpha), and IL-10 were determined along with TLR4 and CD14 expression.

Results: TLR4 expression was similar in patients carrying or not carrying the variant. In contrast, both LPS and HSPB8 resulted in significantly lower secretion of IL-6, TNF-alpha, and IL-10 in those who carried the variant, whereas the frequency of CD14+ cells was higher in these individuals.

Conclusion: TLR4 variant clearly reduces its potency to mediate signaling. Correction for CD14+ cells is necessary in comparable experiments.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Arthritis, Rheumatoid / blood
  • Arthritis, Rheumatoid / genetics*
  • Cytokines / metabolism*
  • Female
  • Gene Expression Regulation*
  • Heat-Shock Proteins / pharmacology
  • Humans
  • Leukocytes, Mononuclear / drug effects
  • Leukocytes, Mononuclear / metabolism
  • Lipopolysaccharides / pharmacology
  • Male
  • Middle Aged
  • Molecular Chaperones
  • Mutation, Missense*
  • Protein Serine-Threonine Kinases / pharmacology
  • Signal Transduction
  • Toll-Like Receptor 4 / genetics*
  • Toll-Like Receptor 4 / metabolism

Substances

  • Cytokines
  • HSPB8 protein, human
  • Heat-Shock Proteins
  • Lipopolysaccharides
  • Molecular Chaperones
  • TLR4 protein, human
  • Toll-Like Receptor 4
  • Protein Serine-Threonine Kinases