L.E.A.P.S. heteroconjugate is able to prevent and treat experimental autoimmune myocarditis by altering trafficking of autoaggressive cells to the heart

Int Immunopharmacol. 2008 May;8(5):624-33. doi: 10.1016/j.intimp.2008.01.004. Epub 2008 Jan 29.

Abstract

We evaluated the efficacy of the Ligand Epitope Antigen Presentation System (L.E.A.P.S.trade mark) in preventing or treating experimental autoimmune myocarditis (EAM) in A/J mice. L.E.A.P.S. (here, J-My-1) is a conjugate of the myocarditogenic peptide of cardiac myosin MyHCalpha(334-352) (My-1) and J peptide, derived from the sequence of human beta-2 microglobulin. Remarkably, early prophylactic (J-My-1 injected on days -14 and -7 before EAM induction), late prophylactic (J-My-1 injected on days 0, 7, 14, and 21), and therapeutic (J-My-1 injected on days 7, 14, and 21 or 10, 17 and 24) administration of J-My-1 significantly decreased the incidence and severity of EAM. However, extended therapeutic treatment was associated with anaphylaxis and death, corresponding with global immune activation associated with J-My-1 treatment. In J-My1-treated animals, we observed expanded numbers of activated CD69+ and CD44+ CD4+ and CD8+ T cells in the spleens. J-My-1 treatment also increased the proportion of CD11c+ dendritic cells in spleens and induced strong production of anti-J-My-1 specific antibodies. J-My-1 injections resulted in decreased levels of chemokines MIP-1alpha and IP-10 in hearts. We propose that J-My-1 treatment interferes with trafficking of autoaggressive immune cells to the heart.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antigen Presentation / drug effects*
  • Autoimmune Diseases / drug therapy*
  • Autoimmune Diseases / pathology
  • Cell Proliferation / drug effects
  • Chemokine CCL3 / biosynthesis
  • Chemokine CXCL10 / biosynthesis
  • Chemokines / biosynthesis
  • Clonal Anergy / drug effects
  • Cytokines / metabolism
  • Dendritic Cells / drug effects
  • Enzyme-Linked Immunosorbent Assay
  • Epitopes / drug effects*
  • Female
  • Histamine Release / drug effects
  • Immunoglobulin J-Chains / pharmacology*
  • Ligands
  • Mice
  • Mice, Inbred A
  • Myocarditis / drug therapy*
  • Myocarditis / pathology
  • Myocardium / metabolism
  • Myocardium / pathology*
  • Spleen / cytology
  • Spleen / drug effects
  • Th1 Cells / drug effects
  • Th2 Cells / drug effects

Substances

  • Chemokine CCL3
  • Chemokine CXCL10
  • Chemokines
  • Cytokines
  • Epitopes
  • Immunoglobulin J-Chains
  • Ligands