Different mechanisms of DEHP-induced hepatocellular adenoma tumorigenesis in wild-type and Ppar alpha-null mice

J Occup Health. 2008;50(2):169-80. doi: 10.1539/joh.l7105.

Abstract

Di (2-ethylhexyl) phthalate (DEHP) exposure is thought to lead to hepatocellular hypertrophy and hyperplasia in rodents mediated via peroxisome proliferator-activated receptor alpha (PPAR alpha). A recent study revealed that long-term exposure to relatively low-dose DEHP (0.05%) caused liver tumors including hepatocellular carcinomas, hepatocellular adenomas, and chologiocellular carcinomas at a higher incidence in Ppar alpha-null mice (25.8%) than in wild-type mice (10.0%). Using tissues with hepatocellular adenoma, microarray (Affymetrix MOE430A) as well as, in part, real-time quantitative PCR analysis was conducted to elucidate the mechanisms of the adenoma formation resulting from DEHP exposure in both genotyped mice. The microarray profiles showed that the up- or down-regulated genes were quite different between hepatocellular adenoma tissues of wild-type and Ppar alpha-null mice exposed to DEHP. The gene expressions of apoptotic peptidase activating factor 1 (Apaf1) and DNA-damage-inducible 45 alpha (Gadd45a) were increased in the hepatocellular adenoma tissues of wild-type mice exposed to DEHP, whereas they were unchanged in corresponding tissues of Ppar alpha-null mice. On the other hand, the expressions of cyclin B2 and myeloid cell leukemia sequence 1 were increased only in the hepatocellular adenoma tissues of Ppar alpha-null mice. Taken together, DEHP may induce hepatocellular adenomas, in part, via suppression of G2/M arrest regulated by Gadd45a and caspase 3-dependent apoptosis in Ppar alpha-null mice, but these genes may not be involved in tumorigenesis in the wild-type mice. In contrast, the expression level of Met was notably increased in the liver adenoma tissue of wild-type mice, which may suggest the involvement of Met in DEHP-induced tumorigenesis in wild-type mice.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Apoptosis / physiology
  • Apoptotic Protease-Activating Factor 1 / antagonists & inhibitors
  • Apoptotic Protease-Activating Factor 1 / biosynthesis
  • Caspase 3 / metabolism
  • Cell Cycle Proteins / antagonists & inhibitors
  • Cell Cycle Proteins / biosynthesis
  • Cell Division / genetics
  • Diethylhexyl Phthalate / administration & dosage
  • Diethylhexyl Phthalate / toxicity*
  • G2 Phase / genetics
  • Gene Expression Profiling
  • Hepatocytes / drug effects
  • Hyperplasia
  • Liver / drug effects*
  • Liver / pathology
  • Liver Neoplasms, Experimental / chemically induced*
  • Liver Neoplasms, Experimental / genetics*
  • Liver Neoplasms, Experimental / pathology
  • Mice
  • Mice, Knockout
  • Microarray Analysis
  • Nuclear Proteins / antagonists & inhibitors
  • Nuclear Proteins / biosynthesis
  • PPAR alpha / deficiency*
  • PPAR alpha / genetics
  • PPAR alpha / metabolism
  • Plasticizers / toxicity
  • Polymerase Chain Reaction
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics

Substances

  • Apaf1 protein, mouse
  • Apoptotic Protease-Activating Factor 1
  • Cell Cycle Proteins
  • Gadd45a protein, mouse
  • Nuclear Proteins
  • PPAR alpha
  • Plasticizers
  • RNA, Messenger
  • Diethylhexyl Phthalate
  • Caspase 3