CD151 accelerates breast cancer by regulating alpha 6 integrin function, signaling, and molecular organization

Cancer Res. 2008 May 1;68(9):3204-13. doi: 10.1158/0008-5472.CAN-07-2949.

Abstract

CD151, a master regulator of laminin-binding integrins (alpha(6)beta(4), alpha(6)beta(1), and alpha(3)beta(1)), assembles these integrins into complexes called tetraspanin-enriched microdomains. CD151 protein expression is elevated in 31% of human breast cancers and is even more elevated in high-grade (40%) and estrogen receptor-negative (45%) subtypes. The latter includes triple-negative (estrogen receptor, progesterone receptor, and HER2 negative) basal-like tumors. CD151 ablation markedly reduced basal-like mammary cell migration, invasion, spreading, and signaling (through FAK, Rac1, and lck) while disrupting epidermal growth factor receptor (EGFR)-alpha(6) integrin collaboration. Underlying these defects, CD151 ablation redistributed alpha(6)beta(4) integrins subcellularly and severed molecular links between integrins and tetraspanin-enriched microdomains. In a prototypical basal-like mammary tumor line, CD151 ablation notably delayed tumor progression in ectopic and orthotopic xenograft models. These results (a) establish that CD151-alpha(6) integrin complexes play a functional role in basal-like mammary tumor progression; (b) emphasize that alpha(6) integrins function via CD151 linkage in the context of tetraspanin-enriched microdomains; and (c) point to potential relevance of CD151 as a high-priority therapeutic target, with relative selectivity (compared with laminin-binding integrins) for pathologic rather than normal physiology.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigens, CD / genetics
  • Antigens, CD / metabolism
  • Antigens, CD / physiology*
  • Breast Neoplasms / genetics*
  • Breast Neoplasms / metabolism
  • Breast Neoplasms / pathology
  • Cell Adhesion / genetics
  • Cell Movement / genetics
  • Disease Progression
  • Epidermal Growth Factor / pharmacology
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Integrin alpha6 / genetics*
  • Integrin alpha6 / metabolism*
  • Integrin alpha6 / physiology
  • Mammary Glands, Human / drug effects
  • Mammary Glands, Human / metabolism
  • Mice
  • Mice, Nude
  • Neoplasm Invasiveness
  • Protein Binding
  • Signal Transduction / genetics
  • Tetraspanin 24
  • Tissue Distribution
  • Transplantation, Heterologous
  • Tumor Cells, Cultured

Substances

  • Antigens, CD
  • CD151 protein, human
  • Cd151 protein, mouse
  • Integrin alpha6
  • Tetraspanin 24
  • Epidermal Growth Factor