Detection of cell-free ERCC1 and thymidylate synthase (TS) mRNA in malignant effusions and its association with anticancer drug sensitivity

Anticancer Res. 2008 Mar-Apr;28(2A):1085-91.

Abstract

Background: The aim of this study was to characterize cell-free mRNA in malignant effusions and evaluate its correlation with the sensitivity of primary tumor cells to cisplatin and 5-fluorouracil (5-FU).

Patients and methods: Malignant effusions were collected from 43 patients and ERCC1 and TS mRNA transcripts in both the supernatants and tumor cells were characterized by real-time quantitative PCR. The sensitivity of primary tumor cells to cisplatin and 5-FU was analyzed using an ATP-TCA assay.

Results: Cell-free ERCC1 and TS mRNA transcripts were observed in 42 out of 43 specimens, with variable levels comparing gene expression patterns in paired-tumor cells (p < 0.0001, p = 0.02, respectively). TS mRNA levels in the supernatants were inversely correlated with the in vitro sensitivity of cancer cells to 5-FU in the gastrointestinal group (p = 0.002).

Conclusion: The cell-free mRNA transcripts in malignant effusions were highly detectable and cell-free TS mRNA in gastrointestinal cancer patients were strongly associated with the sensitivity of primary cancer cells to 5-FU in vitro.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Ascites / metabolism*
  • Cell-Free System
  • Cisplatin / therapeutic use
  • DNA-Binding Proteins / genetics*
  • Drug Resistance, Neoplasm
  • Endonucleases / genetics*
  • Female
  • Fluorouracil / therapeutic use
  • Humans
  • Male
  • Middle Aged
  • Pleural Effusion, Malignant / chemistry*
  • RNA, Messenger / analysis
  • Thymidylate Synthase / genetics*

Substances

  • DNA-Binding Proteins
  • RNA, Messenger
  • Thymidylate Synthase
  • ERCC1 protein, human
  • Endonucleases
  • Cisplatin
  • Fluorouracil