Cell-penetrating peptide TP10 shows broad-spectrum activity against both Plasmodium falciparum and Trypanosoma brucei brucei

Antimicrob Agents Chemother. 2008 Sep;52(9):3414-7. doi: 10.1128/AAC.01450-07. Epub 2008 Jun 2.

Abstract

Malaria and trypanosomiasis are diseases which afflict millions and for which novel therapies are urgently required. We have tested two well-characterized cell-penetrating peptides (CPPs) for antiparasitic activity. One CPP, designated TP10, has broad-spectrum antiparasitic activity against Plasmodium falciparum, both blood and mosquito stages, and against blood-stage Trypanosoma brucei brucei.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antimalarials / pharmacology*
  • Cell Membrane / metabolism*
  • Humans
  • Molecular Sequence Data
  • Parasitic Sensitivity Tests
  • Peptides / chemistry
  • Peptides / pharmacology*
  • Peptides / therapeutic use
  • Plasmodium falciparum / drug effects*
  • Plasmodium falciparum / growth & development
  • Trypanocidal Agents / pharmacology*
  • Trypanosoma brucei brucei / drug effects*
  • Trypanosoma brucei brucei / growth & development

Substances

  • Antimalarials
  • Peptides
  • Trypanocidal Agents