Synthesis and antiinflammatory activity of indole carboxylic acids and esters

Acta Pharm Nord. 1991;3(1):5-8.

Abstract

1-Phenylalkylindole-3-carboxylic acids 1-4, indole-1-acetic acids/esters 5-10 and the hydrazones 11-15 were prepared and submitted to the rat paw edema test using carrageenin. In the first two groups of compounds, the 2-chloro indoles were more active than the corresponding indole derivatives. In the third group the activity seemed to be determined largely by the substituent at the 1-position.

MeSH terms

  • Anti-Inflammatory Agents, Non-Steroidal / chemical synthesis
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology
  • Carboxylic Acids / chemical synthesis
  • Carboxylic Acids / pharmacology
  • Esters / chemical synthesis
  • Esters / pharmacology
  • Indoles / chemical synthesis*
  • Indoles / pharmacology

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Carboxylic Acids
  • Esters
  • Indoles