Smad2 functions as a co-activator of canonical Wnt/beta-catenin signaling pathway independent of Smad4 through histone acetyltransferase activity of p300

Cell Signal. 2008 Sep;20(9):1632-41. doi: 10.1016/j.cellsig.2008.05.003. Epub 2008 May 18.

Abstract

Both canonical Wnt/beta-catenin and TGFbeta/Smad signaling pathways coordinately regulate pattern formation during embryogenesis as well as tumor progression. Evidence of cross-talk between these two pathways has been reported. Here we demonstrated that the Activin-like kinase 4 (Alk4)/Smad2 pathway facilitates the transcriptional activity of the oncogenic Wnt/beta-catenin/Tcf4 pathway through a novel Smad4-independent mechanism. Upon activation, Smad2 physically interacted with Tcf4, beta-catenin and the co-activator p300 to enhance transcriptional activity of beta-catenin/Tcf4 through the histone acetyltransferase activity of p300. Transactivation by Smad2 was independent of a Smad-binding element (SBE) and Smad4. Indeed, the enhancement of beta-catenin/Tcf4 transcriptional activity by activated Smad2 was negatively regulated by the presence of Smad4. Moreover, a tumor-derived missense mutant of Smad2, lacking the ability to bind to Smad4 was still able to enhance the Tcf4 transcriptional reporter in the presence of beta-catenin and Tcf4. Our findings suggest that Smad2 may function as an activator of canonical Wnt/beta-catenin/Tcf4 signaling through a SBE/Smad4-independent pathway.

Publication types

  • Research Support, N.I.H., Intramural

MeSH terms

  • Activin Receptors, Type I / metabolism
  • Cell Line
  • Histone Acetyltransferases / metabolism*
  • Humans
  • Models, Genetic
  • Protein Binding
  • Signal Transduction*
  • Smad2 Protein / genetics
  • Smad2 Protein / metabolism*
  • Smad4 Protein / metabolism
  • TCF Transcription Factors / metabolism
  • Transcription Factor 7-Like 2 Protein
  • Transcription, Genetic
  • Transcriptional Activation
  • Wnt Proteins / metabolism*
  • beta Catenin / metabolism*
  • p300-CBP Transcription Factors / metabolism*

Substances

  • Smad2 Protein
  • Smad4 Protein
  • TCF Transcription Factors
  • TCF7L2 protein, human
  • Transcription Factor 7-Like 2 Protein
  • Wnt Proteins
  • beta Catenin
  • Histone Acetyltransferases
  • p300-CBP Transcription Factors
  • Activin Receptors, Type I