Role of microsomal prostaglandin E synthase-1 (mPGES1)-derived PGE2 in patency of the ductus arteriosus in the mouse

Pediatr Res. 2008 Nov;64(5):523-7. doi: 10.1203/PDR.0b013e318184d29c.

Abstract

Prostaglandin E2 (PGE2) plays a key role in the ductus arteriosus, prenatally by maintaining patency and postnatally by promoting tissue remodeling for closure. Here, by using near-term mouse fetuses with (wild-type, WT) and without microsomal PGE synthase-1 (mPGES1-/-), we have examined the importance of this enzyme for PGE2 formation and function. mPGES1-/- ductus, unlike WT ductus, contracted little, or not all, to indomethacin in vitro. Coincidentally, as evident from responses to NG-nitro-L-arginine methyl ester and zinc photoporphyrin, the mutant showed no significant enhancement of nitric oxide (NO)- and carbon monoxide (CO)-based relaxation. mPGES1 suppression differs, therefore, from cyclooxygenase (COX) suppression, whether genetically or pharmacologically induced, where NO is markedly up-regulated. In vivo, the ductus was patent, albeit occasionally with a narrowed lumen, in all mPGES1-/- fetuses. Conversely, postnatal closure progressed regularly in mPGES1-/- animals thanks to residual PGE2 originating via mPGES2. We conclude that mPGES1 is critical for PGE2 formation in the ductus but its loss does not entail compensatory up-regulation of other relaxing mechanisms. Accordingly, an mPGES1 inhibitor stands out as a prospective better tool, compared with the currently used COX inhibitors, for the management of premature infants with persistent ductus.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carbon Monoxide / metabolism
  • Cyclooxygenase Inhibitors / pharmacology
  • Dinoprostone / metabolism*
  • Ductus Arteriosus / enzymology*
  • Ductus Arteriosus / physiopathology
  • Ductus Arteriosus, Patent / enzymology*
  • Ductus Arteriosus, Patent / physiopathology
  • Enzyme Inhibitors / pharmacology
  • Gestational Age
  • Heme Oxygenase (Decyclizing) / antagonists & inhibitors
  • Heme Oxygenase (Decyclizing) / metabolism
  • Indomethacin / pharmacology
  • Intramolecular Oxidoreductases / deficiency
  • Intramolecular Oxidoreductases / genetics
  • Intramolecular Oxidoreductases / metabolism*
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • NG-Nitroarginine Methyl Ester / pharmacology
  • Nitric Oxide / metabolism
  • Nitric Oxide Synthase / antagonists & inhibitors
  • Nitric Oxide Synthase / metabolism
  • Prostaglandin-E Synthases
  • Protoporphyrins / pharmacology
  • RNA, Messenger / metabolism
  • Vascular Patency*

Substances

  • Cyclooxygenase Inhibitors
  • Enzyme Inhibitors
  • Protoporphyrins
  • RNA, Messenger
  • zinc protoporphyrin
  • Nitric Oxide
  • Carbon Monoxide
  • Nitric Oxide Synthase
  • Heme Oxygenase (Decyclizing)
  • Intramolecular Oxidoreductases
  • Prostaglandin-E Synthases
  • Ptges protein, mouse
  • Dinoprostone
  • NG-Nitroarginine Methyl Ester
  • Indomethacin