Catalytic activity of nuclear PLC-beta(1) is required for its signalling function during C2C12 differentiation

Cell Signal. 2008 Nov;20(11):2013-21. doi: 10.1016/j.cellsig.2008.07.009. Epub 2008 Jul 20.

Abstract

Here we report that PLC-beta(1) catalytic activity plays a role in the increase of cyclin D3 levels and induces the differentiation of C2C12 skeletal muscle cells. PLC-beta(1) mutational analysis revealed the importance of His(331) and His(378) for the catalysis. The expression of PLC-beta(1) and cyclin D3 proteins is highly induced during the process of skeletal myoblast differentiation. We have previously shown that PLC-beta(1) activates cyclin D3 promoter during the differentiation of myoblasts to myotubes, indicating that PLC-beta(1) is a crucial regulator of the mouse cyclin D3 gene. We show that after insulin treatment cyclin D3 mRNA levels are lower in cells overexpressing the PLC-beta(1) catalytically inactive form in comparison to wild type cells. We describe a novel signalling pathway elicited by PLC-beta(1) that modulates AP-1 activity. Gel mobility shift assay and supershift performed with specific antibodies indicate that the c-jun binding site is located in a cyclin D3 promoter region specifically regulated by PLC-beta(1) and that c-Jun binding activity is significantly increased by insulin and PLC-beta(1) overexpression. Mutation of AP-1 site decreased the basal cyclin D3 promoter activity and eliminated its induction by insulin and PLC-beta(1). These results hint at the fact that PLC-beta(1) catalytic activity signals a c-jun/AP-1 target gene, i.e. cyclin D3, during myogenic differentiation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Biocatalysis / drug effects
  • Cell Differentiation* / drug effects
  • Cell Nucleus / drug effects
  • Cell Nucleus / enzymology*
  • Cyclin D3
  • Cyclins / genetics
  • Gene Expression Profiling
  • Insulin / pharmacology
  • Lipase / metabolism
  • Mice
  • Molecular Sequence Data
  • Muscle Development / drug effects
  • Mutagenesis / drug effects
  • Mutant Proteins / metabolism
  • Mutation / genetics
  • Myoblasts / cytology*
  • Myoblasts / drug effects
  • Myoblasts / enzymology*
  • NF-kappa B / metabolism
  • Phospholipase C beta / chemistry
  • Phospholipase C beta / metabolism*
  • Promoter Regions, Genetic
  • Protein Transport / drug effects
  • Proto-Oncogene Proteins c-jun / metabolism
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Rats
  • Signal Transduction* / drug effects
  • Transcription, Genetic / drug effects

Substances

  • CCND3 protein, human
  • Ccnd3 protein, mouse
  • Ccnd3 protein, rat
  • Cyclin D3
  • Cyclins
  • Insulin
  • Mutant Proteins
  • NF-kappa B
  • Proto-Oncogene Proteins c-jun
  • RNA, Messenger
  • Lipase
  • Phospholipase C beta