Cadmium activates the mitogen-activated protein kinase (MAPK) pathway via induction of reactive oxygen species and inhibition of protein phosphatases 2A and 5

Free Radic Biol Med. 2008 Oct 1;45(7):1035-44. doi: 10.1016/j.freeradbiomed.2008.07.011. Epub 2008 Jul 26.

Abstract

Cadmium (Cd), a highly toxic environmental pollutant, induces neurodegenerative diseases. Recently we have demonstrated that Cd may induce neuronal apoptosis in part through activation of c-Jun N-terminal kinase (JNK) and extracellular signal-regulated kinase 1/2 (Erk1/2) pathways. However, the underlying mechanism remains enigmatic. Here we show that Cd induced generation of reactive oxygen species (ROS), leading to apoptosis of PC12 and SH-SY5Y cells. Pretreatment with N-acetyl-L-cysteine (NAC) scavenged Cd-induced ROS, and prevented cell death, suggesting that Cd-induced apoptosis is attributed to its induction of ROS. Furthermore, we found that Cd-induced ROS inhibited serine/threonine protein phosphatases 2A (PP2A) and 5 (PP5), leading to activation of Erk1/2 and JNK, which was abrogated by NAC. Overexpression of PP2A or PP5 partially prevented Cd-induced activation of Erk1/2 and JNK, as well as cell death. Cd-induced ROS was also linked to the activation of caspase-3. Pretreatment with inhibitors of JNK (SP600125) and Erk1/2 (U0126) partially blocked Cd-induced cleavage of caspase-3 and prevented cell death. However, zVAD-fmk, a pan caspase inhibitor, only partially prevented Cd-induced apoptosis. The results indicate that Cd induction of ROS inhibits PP2A and PP5, leading to activation of JNK and Erk1/2 pathways, and consequently resulting in caspase-dependent and -independent apoptosis of neuronal cells. The findings strongly suggest that the inhibitors of JNK, Erk1/2, or antioxidants may be exploited for prevention of Cd-induced neurodegenerative diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcysteine / pharmacology
  • Animals
  • Apoptosis / drug effects
  • Blotting, Western
  • Cadmium / toxicity*
  • Cell Line, Tumor
  • Enzyme Activation / drug effects
  • Enzyme Inhibitors / pharmacology
  • Flow Cytometry
  • Free Radical Scavengers / pharmacology
  • Humans
  • Mitogen-Activated Protein Kinases / drug effects*
  • Nuclear Proteins / drug effects*
  • Phosphoprotein Phosphatases / drug effects*
  • Protein Phosphatase 2 / drug effects*
  • Rats
  • Reactive Oxygen Species / metabolism*
  • Signal Transduction / drug effects*

Substances

  • Enzyme Inhibitors
  • Free Radical Scavengers
  • Nuclear Proteins
  • Reactive Oxygen Species
  • Cadmium
  • Mitogen-Activated Protein Kinases
  • Phosphoprotein Phosphatases
  • Protein Phosphatase 2
  • protein phosphatase 5
  • Acetylcysteine