[Effect of decitabine combined with Trichostatin A on MDS cell line SKM-1 in vitro]

Zhongguo Shi Yan Xue Ye Xue Za Zhi. 2008 Aug;16(4):819-23.
[Article in Chinese]

Abstract

The study was purposed to explore the effect and mechanisms of decitabine and/or Trichostatin A (TSA) on SKM-1 cells in vitro. The effect of decitabine and/or TSA on proliferation of SKM-1cells was analyzed with trypan blue exclusion; the differentiation of SKM-1 cells was detected by nitro-blue tetrazolium (NBT) reduction and flow cytometry; the apoptosis of cells was measured by Annexin V-FITC; the mRNA expression of Fas, survivin and P15(INK4B) in cells treated with decitabine and/or TSA was evaluated by RT-PCR. The results showed that decitabine and/or TSA were capable of inhibiting SKM-1 cell growth and promoting cell differentiation; they stimulated the expression of CD14 and CD11b and inhibited HLA-DR expression; meanwhile and decitabine or/and TSA could induce cell apoptosis, up-regulate mRNA expression of Fas and P15(INK4B), and down-regulate survivin mRNA expression. It is concluded that decitabine can induce apoptosis/differentiation of SKM-1 cells, whose mechanisms may related to the expression of Fas, survivin and P15(INK4B). Decitabine has the synergistic effect with TSA.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antimetabolites, Antineoplastic / pharmacology
  • Apoptosis / drug effects*
  • Azacitidine / analogs & derivatives*
  • Azacitidine / pharmacology
  • Cell Differentiation
  • Cell Line, Tumor
  • Cell Proliferation / drug effects*
  • Decitabine
  • Drug Synergism
  • Humans
  • Hydroxamic Acids / pharmacology*
  • Inhibitor of Apoptosis Proteins
  • Microtubule-Associated Proteins / genetics
  • Microtubule-Associated Proteins / metabolism
  • Myelodysplastic Syndromes / pathology*
  • Survivin
  • fas Receptor / genetics
  • fas Receptor / metabolism

Substances

  • Antimetabolites, Antineoplastic
  • BIRC5 protein, human
  • Hydroxamic Acids
  • Inhibitor of Apoptosis Proteins
  • Microtubule-Associated Proteins
  • Survivin
  • fas Receptor
  • trichostatin A
  • Decitabine
  • Azacitidine