Cdk5 phosphorylates Cdh1 and modulates cyclin B1 stability in excitotoxicity

EMBO J. 2008 Oct 22;27(20):2736-45. doi: 10.1038/emboj.2008.195. Epub 2008 Sep 25.

Abstract

Anaphase-promoting complex/cyclosome (APC/C), an E3 ubiquitin ligase that destabilizes cell cycle proteins, is activated by Cdh1 in post-mitotic neurons, where it regulates axonal growth, synaptic plasticity and survival. The APC/C-Cdh1 substrate, cyclin B1, has been found to accumulate in degenerating brain areas in Alzheimer's disease and stroke. This highlights the importance of elucidating cyclin B1 regulation by APC/C-Cdh1 in neurons under stress conditions relevant to neurological disease. Here, we report that stimulation of N-methyl-D-aspartate receptors (NMDARs) that occurs in neurodegenerative diseases promoted the accumulation of cyclin B1 in the nuclei of cortical neurons; this led the neurons to undergo apoptotic death. Moreover, we found that the Ser-40, Thr-121 and Ser-163 triple phosphorylation of Cdh1 by the cyclin-dependent kinase-5 (Cdk5)-p25 complex was necessary and sufficient for cyclin B1 stabilization and apoptotic death after NMDAR stimulation. These results reveal Cdh1 as a novel Cdk5 substrate that mediates cyclin B1 neuronal accumulation in excitotoxicity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis
  • Cadherins / metabolism*
  • Cell Nucleus / metabolism
  • Cells, Cultured
  • Cyclin B / metabolism*
  • Cyclin B1
  • Cyclin-Dependent Kinase 5 / metabolism*
  • Models, Biological
  • Neurons / metabolism
  • Phosphorylation
  • Plasmids / metabolism
  • Rats
  • Rats, Wistar
  • Receptors, N-Methyl-D-Aspartate / metabolism
  • Serine / chemistry

Substances

  • Cadherins
  • Ccnb1 protein, rat
  • Cyclin B
  • Cyclin B1
  • Receptors, N-Methyl-D-Aspartate
  • Serine
  • Cyclin-Dependent Kinase 5