In situ gel based on gellan gum as new carrier for nasal administration of mometasone furoate

Int J Pharm. 2009 Jan 5;365(1-2):109-15. doi: 10.1016/j.ijpharm.2008.08.042. Epub 2008 Sep 7.

Abstract

The main purpose of this study was to prepare a novel in situ gel system for nasal delivery of MF and study its efficacy on allergic rhinitis model. An ion-activated in situ gel was developed and characterized with gellan gum as a carrier. The system was stable kept at 40+/-2 degrees C for 6 months, and the micrographic results showed that in situ gel was safety without mucosa irritation when given at 20 microg once daily for 1 month to rats with allergic rhinitis. MF in gellan gum produced obviously effect on allergic rhinitis at the doses of 20 microg/body following intranasal administration, and the efficacy was significantly superior to that of the common suspension (P<0.01). The in situ gel system is a promising approach for the intranasal delivery of MF for the therapeutic effects improvement.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Intranasal
  • Animals
  • Anti-Allergic Agents / administration & dosage*
  • Anti-Allergic Agents / toxicity
  • Anura
  • Disease Models, Animal
  • Drug Carriers / chemistry
  • Drug Stability
  • Drug Storage
  • Female
  • Gels
  • Male
  • Mometasone Furoate
  • Nasal Mucosa / drug effects
  • Nasal Mucosa / metabolism
  • Polysaccharides, Bacterial / chemistry*
  • Pregnadienediols / administration & dosage*
  • Pregnadienediols / toxicity
  • Rats
  • Rats, Wistar
  • Rhinitis, Allergic, Perennial / drug therapy*
  • Toxicity Tests

Substances

  • Anti-Allergic Agents
  • Drug Carriers
  • Gels
  • Polysaccharides, Bacterial
  • Pregnadienediols
  • Mometasone Furoate
  • gellan gum