Anticancer effect of celecoxib via COX-2 dependent and independent mechanisms in human gastric cancers cells

Dig Dis Sci. 2009 Jul;54(7):1418-24. doi: 10.1007/s10620-008-0510-9. Epub 2008 Oct 16.

Abstract

Cyclooxygenase-2 (COX-2) inhibitors cause growth inhibition of human gastric carcinoma cells, but it remains unclear whether this is both COX-2 dependent and independent. The related mechanisms remain to be determined. Both low COX-2 expressing gastric carcinoma and high COX-2 expressing gastric carcinoma cells were used to study the effect and mechanisms of celecoxib on gastric carcinoma cell growth. Celecoxib resulted in comparable growth inhibition in AGS cells with stable transfections of small interfering RNA (siRNA) against COX-2 (SAC) and negative control vector (NC) cells. Simultaneously, celecoxib resulted in significant reduction of Bcl-2 and significant increase of p21(WAF1) and p27(KIP1) in SAC and NC cells. The present study shows that celecoxib causes growth inhibition of gastric carcinoma cells by decreasing Bcl-2 of cyclooxygenase-2-dependent pathway, and by increasing p21(WAF1) and p27(KIP1) of cyclooxygenase-2-independent pathway. These data extend our knowledge on the effect and mechanisms of celecoxib-induced inhibition of gastric carcinoma cell growth.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blotting, Western
  • Celecoxib
  • Cell Proliferation / drug effects
  • Chemoprevention
  • Colony-Forming Units Assay
  • Cyclin-Dependent Kinase Inhibitor p21 / metabolism
  • Cyclin-Dependent Kinase Inhibitor p21 / physiology
  • Cyclin-Dependent Kinase Inhibitor p27 / metabolism
  • Cyclooxygenase 2 / metabolism*
  • Cyclooxygenase 2 Inhibitors / pharmacology*
  • Genes, bcl-2 / physiology
  • Humans
  • Pyrazoles / pharmacology*
  • RNA, Small Interfering / drug effects
  • Reverse Transcriptase Polymerase Chain Reaction
  • Stomach Neoplasms / drug therapy
  • Stomach Neoplasms / physiopathology*
  • Stomach Neoplasms / prevention & control
  • Sulfonamides / pharmacology*
  • Tumor Cells, Cultured

Substances

  • CDKN1A protein, human
  • Cyclin-Dependent Kinase Inhibitor p21
  • Cyclooxygenase 2 Inhibitors
  • Pyrazoles
  • RNA, Small Interfering
  • Sulfonamides
  • Cyclin-Dependent Kinase Inhibitor p27
  • Cyclooxygenase 2
  • Celecoxib