Activation of beta-Catenin in mouse prostate causes HGPIN and continuous prostate growth after castration

Prostate. 2009 Feb 15;69(3):249-62. doi: 10.1002/pros.20877.

Abstract

Background: The role of Wnt/beta-Catenin signaling in embryogenesis and carcinogenesis has been extensively studied in organs such as colon, lung and pancreas, but little is known about Wnt/beta-Catenin signaling in the prostate. Although stabilizing mutations in APC and beta-Catenin are rare in primary prostate tumors, recent studies suggest that cytoplasmic/nuclear beta-Catenin is associated with advanced, metastatic, hormone-refractory prostate carcinoma.

Methods: To better understand the role of beta-Catenin in prostatic development and carcinogenesis, we studied Wnt expression during prostate development and activated Wnt/beta-Catenin signaling in the developing and adult prostate.

Results: Our results demonstrated that during prostate development Wnt ligands display a dynamic expression pattern. Activation of beta-Catenin during prostate development caused epithelial hyperplasia followed by prostatic intraepithelial neoplasia (PIN) in prostate. In the adult prostate, activation of beta-Catenin resulted in high grade PIN (HGPIN) and continuous prostatic growth after castration. As a result of activation of beta-Catenin, AR was first up-regulated with the emergence of epithelial hyperplasia, but was later down-regulated when HGPIN developed. Furthermore, activation of beta-Catenin induced Foxa2 re-expression in adult prostate which normally is only expressed in the embryonic budding stage during prostate development.

Conclusions: The results from this study strongly suggest that Wnt/beta-Catenin signaling is involved in the regulation of prostate development and confirm that constitutive activation of this pathway enables the mouse prostate to grow after castration.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Age Factors
  • Androgens / metabolism
  • Animals
  • Female
  • Gene Expression Regulation, Developmental
  • Gene Expression Regulation, Neoplastic
  • Hepatocyte Nuclear Factor 3-beta / genetics
  • Hepatocyte Nuclear Factor 3-beta / metabolism
  • Homeodomain Proteins / genetics
  • Integrases / genetics
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Mutant Strains
  • Mice, Nude
  • Orchiectomy*
  • Pregnancy
  • Prostate / growth & development
  • Prostate / physiology*
  • Prostatic Intraepithelial Neoplasia / physiopathology*
  • Prostatic Neoplasms / physiopathology*
  • Signal Transduction / physiology
  • Transcription Factors / genetics
  • Wnt Proteins / metabolism
  • beta Catenin / genetics
  • beta Catenin / metabolism*

Substances

  • Androgens
  • CTNNB1 protein, mouse
  • Foxa2 protein, mouse
  • Homeodomain Proteins
  • Nkx3-1 protein, mouse
  • Transcription Factors
  • Wnt Proteins
  • beta Catenin
  • Hepatocyte Nuclear Factor 3-beta
  • Cre recombinase
  • Integrases