Peroxisome proliferator-activated receptor gamma overexpression and knockdown: impact on human B cell lymphoma proliferation and survival

Cancer Immunol Immunother. 2009 Jul;58(7):1071-83. doi: 10.1007/s00262-008-0625-z. Epub 2008 Nov 19.

Abstract

Peroxisome proliferator-activated receptor gamma (PPARgamma) is a multifunctional transcription factor that regulates adipogenesis, immunity and inflammation. Our laboratory previously demonstrated that PPARgamma ligands induce apoptosis in malignant B cells. While malignant B lineage cells such as B cell lymphoma express PPARgamma, its physiological function remains unknown. Herein, we demonstrate that silencing PPARgamma expression by RNAi in human Burkitt's type B lymphoma cells increased basal and mitogen-induced proliferation and survival, which was accompanied by enhanced NF-kappaB activity and increased expression of Bcl-2. These cells also had increased survival upon exposure to PPARgamma ligands and exhibited a less differentiated phenotype. In contrast, PPARgamma overexpression in B lymphoma cells inhibited cell growth and decreased their proliferative response to mitogenic stimuli. These cells were also more sensitive to PPARgamma-ligand induced growth arrest and displayed a more differentiated phenotype. Collectively, these findings support a regulatory role for PPARgamma in the proliferation, survival and differentiation of malignant B cells. These findings further suggest the potential of PPARgamma as a therapeutic target for B cell malignancy.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Burkitt Lymphoma / genetics
  • Burkitt Lymphoma / pathology*
  • Cell Line, Tumor
  • Cell Proliferation
  • Cell Survival
  • Gene Knockdown Techniques
  • Genetic Vectors / metabolism
  • Humans
  • Ligands
  • NF-kappa B / metabolism*
  • PAX5 Transcription Factor / metabolism*
  • PPAR gamma / genetics
  • PPAR gamma / metabolism*
  • Positive Regulatory Domain I-Binding Factor 1
  • Proto-Oncogene Proteins c-bcl-2 / metabolism*
  • RNA Interference
  • Repressor Proteins / metabolism*

Substances

  • Ligands
  • NF-kappa B
  • PAX5 Transcription Factor
  • PAX5 protein, human
  • PPAR gamma
  • Proto-Oncogene Proteins c-bcl-2
  • Repressor Proteins
  • PRDM1 protein, human
  • Positive Regulatory Domain I-Binding Factor 1