Activation of mTOR in a subgroup of ovarian carcinomas: correlation with p-eIF-4E and prognosis

Oncol Rep. 2008 Dec;20(6):1409-17.

Abstract

Ovarian carcinoma patients have an extremely poor prognosis; therefore, new molecular therapeutic approaches are urgently needed. The mTOR pathway, which may be targeted by substances such as Rapamycin or RAD001, is emerging as a promising target for anticancer therapy. So far, the expression and prognostic impact of mTOR signalling elements have not been completely studied in ovarian tumors. We analyzed p-mTOR, p-4E-BP1 and p-eIF-4E in 107 human ovarian lesions and observed an overexpression of p-mTOR (47%) and p-eIF-4E (56%) protein in primary ovarian carcinomas as compared to borderline tumors. Phospho-mTOR expression was significantly related to p-eIF-4E (p< or =0.001) and serous histological type (p=0.03). Increased p-4E-BP1 (31%) was associated with poor differentiation (p=0.04) and higher mitotic rate (p=0.004). In univariate analysis, increased expression of p-mTOR and p-eIF-4E was significantly associated with better overall survival (p=0.003, p=0.029). To connect the expression data with mechanistic studies, a set of 10 ovarian cancer cell lines was used. Expression of p-mTOR was increased in all cancer cell lines as compared to ovarian surface epithelial (HOSE) cells. Rapamycin treatment revealed a reduction of p-mTOR and p-4E-BP1 but increased p-AKT levels. We show for the first time an association of p-mTOR and p-eIF-4E with better overall survival for ovarian cancer patients. The combined results of our in vivo and cell culture studies suggest that a subpopulation of these patients may benefit from mTOR inhibition. The design of future clinical trials should incorporate biomarker testing to determine predictive markers for response to mTOR inhibitors.

MeSH terms

  • Aged
  • Apoptosis
  • Cell Cycle
  • Cell Line, Tumor
  • Enzyme Activation
  • Eukaryotic Initiation Factor-4E / biosynthesis*
  • Eukaryotic Initiation Factor-4E / physiology*
  • Female
  • Gene Expression Profiling
  • Humans
  • Immunohistochemistry / methods
  • Middle Aged
  • Mitosis
  • Ovarian Neoplasms / metabolism*
  • Prognosis
  • Protein Kinases / biosynthesis*
  • Protein Kinases / physiology*
  • TOR Serine-Threonine Kinases

Substances

  • Eukaryotic Initiation Factor-4E
  • Protein Kinases
  • MTOR protein, human
  • TOR Serine-Threonine Kinases