Complete NMR assignment and absolute configuration of feronielloside, a new acetylcholinesterase inhibitor from Feroniella lucida

Nat Prod Res. 2008;22(15):1297-303. doi: 10.1080/14786410801980626.

Abstract

Feronielloside (1), a new furanocoumarin glycoside, was isolated from roots of Feroniella lucida. The structure of 1 was elucidated by combined spectroscopic and chemical analysis. The absolute configuration of the chiral center in geranyl-derived side chain was confirmed by modified Mosher's method. Feronielloside inhibited acetylcholinesterase with IC(50) value of 24.7 mM.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholinesterase / metabolism*
  • Cholinesterase Inhibitors* / chemistry
  • Cholinesterase Inhibitors* / isolation & purification
  • Cholinesterase Inhibitors* / pharmacology
  • Coumarins* / chemistry
  • Coumarins* / isolation & purification
  • Coumarins* / pharmacology
  • Furans* / chemistry
  • Furans* / isolation & purification
  • Furans* / pharmacology
  • Glycosides* / chemistry
  • Glycosides* / isolation & purification
  • Glycosides* / pharmacology
  • Molecular Structure
  • Nuclear Magnetic Resonance, Biomolecular
  • Plant Roots / chemistry
  • Plants, Medicinal / chemistry*
  • Rutaceae / chemistry*
  • Thailand

Substances

  • Cholinesterase Inhibitors
  • Coumarins
  • Furans
  • Glycosides
  • feronielloside
  • Acetylcholinesterase