Cognitive and cerebral metabolic effects of celecoxib versus placebo in people with age-related memory loss: randomized controlled study

Am J Geriatr Psychiatry. 2008 Dec;16(12):999-1009. doi: 10.1097/JGP.0b013e31818cd3a4.

Abstract

Objective: Because anti-inflammatory drugs may delay cognitive decline and influence brain metabolism in normal aging, the authors determined the effects of the cyclooxygenase-2 inhibitor, celecoxib, on cognitive performance and regional cerebral glucose metabolism in nondemented volunteers with mild age-related memory decline.

Design: Randomized, double-blind, placebo-controlled, parallel group trial with 18-months of exposure to study medication.

Setting: University research institute.

Participants: Eighty-eight subjects, aged 40-81 years (mean: 58.7, SD: 8.9 years) with mild self-reported memory complaints but normal memory performance scores were recruited from community physician referrals, media coverage, and advertising. Forty subjects completed the study.

Interventions: Daily celecoxib dose of 200 or 400 mg, or placebo.

Main outcome measures: Standardized neuropsychological test battery and statistical parametric mapping (SPM) of FDG-PET scans performed during mental rest.

Results: Measures of cognition showed significant between-group differences in executive functioning (F [1, 30] = 5.06, p = 0.03) and language/semantic memory (F [1, 31] = 6.19, p = 0.02), favoring the celecoxib group compared with the placebo group. Concomitantly, FDG-PET scans demonstrated bilateral metabolic increases in prefrontal cortex in the celecoxib group in the vicinity of Brodmann's areas 9 and 10, but not in the placebo group. SPM analyses of the PET data pooled by treatment arm corresponded to a 6% increase in activity over pretreatment levels (p <0.01, after adjustment for multiple comparisons).

Conclusions: These results suggest that daily celecoxib use may improve cognitive performance and increase regional brain metabolism in people with age-associated memory decline.

Publication types

  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Adult
  • Age Factors
  • Aged
  • Aged, 80 and over
  • Anti-Inflammatory Agents, Non-Steroidal / metabolism
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Apolipoprotein E4 / genetics
  • Apolipoprotein E4 / metabolism
  • Celecoxib
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / metabolism
  • Cognition Disorders / drug therapy*
  • Cognition Disorders / metabolism
  • Cyclooxygenase 2 Inhibitors / metabolism
  • Cyclooxygenase 2 Inhibitors / pharmacology
  • Cyclooxygenase 2 Inhibitors / therapeutic use*
  • Double-Blind Method
  • Female
  • Fluorodeoxyglucose F18 / metabolism
  • Fluorodeoxyglucose F18 / pharmacology
  • Humans
  • Male
  • Memory Disorders / drug therapy*
  • Memory Disorders / metabolism*
  • Middle Aged
  • Neuropsychological Tests
  • Positron-Emission Tomography
  • Pyrazoles / administration & dosage
  • Pyrazoles / adverse effects
  • Pyrazoles / therapeutic use*
  • Radiopharmaceuticals
  • Sulfonamides / administration & dosage
  • Sulfonamides / adverse effects
  • Sulfonamides / therapeutic use*
  • Treatment Outcome

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Apolipoprotein E4
  • Cyclooxygenase 2 Inhibitors
  • Pyrazoles
  • Radiopharmaceuticals
  • Sulfonamides
  • Fluorodeoxyglucose F18
  • Celecoxib

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