Immunostimulation and anti-DNA antibody production by backbone modified CpG-DNA

Biochem Biophys Res Commun. 2009 Feb 6;379(2):362-7. doi: 10.1016/j.bbrc.2008.12.063. Epub 2008 Dec 25.

Abstract

Oligodeoxynucleotides containing immunostimulatory CpG motifs (CpG-DNA) have gained attention as potentially useful therapeutics. However, the phosphorothioate-modified CpG-DNAs (PS-ODN) can induce backbone-related side effects. Here, we compared the immunostimulatory activity of natural phosphodiester CpG-DNA (PO-ODN) from Mycobacterium bovis and PS-ODN in mice. Both PO-ODN and PS-ODN induced production of IL-12. PS-ODN increased spleen weights, spleen cell numbers, and the migration of macrophages into the peritoneal cavity in the mice in a CG sequence-dependent manner. PS-ODN induced anti-PS-ODN antibody production in the mice, and the PS-ODN-specific IgM was cross-reactive with other PS-ODNs in a CG sequence-independent manner. In contrast, PO-ODN did not affect on spleen weights, cell numbers, or IgM production. These results may provide an explanation for the side effects in immunotherapeutic application of PS-ODN. They also suggest that PO-ODN may be more optimal than PS-ODN to enhance innate immune responses without severe side effects.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Antinuclear / biosynthesis*
  • Antibodies, Antinuclear / immunology
  • Cell Movement
  • CpG Islands / immunology*
  • DNA / immunology*
  • DNA / pharmacology
  • Immunization
  • Interleukin-12 / immunology
  • Macrophages, Peritoneal / drug effects
  • Macrophages, Peritoneal / immunology
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Mycobacterium bovis / genetics
  • Mycobacterium bovis / immunology
  • Phosphorothioate Oligonucleotides / immunology*
  • Phosphorothioate Oligonucleotides / pharmacology
  • Splenomegaly / immunology*

Substances

  • Antibodies, Antinuclear
  • Phosphorothioate Oligonucleotides
  • Interleukin-12
  • DNA