Nebulized phosphodiesterase III inhibitor during warm ischemia attenuates pulmonary ischemia-reperfusion injury

J Heart Lung Transplant. 2009 Jan;28(1):79-84. doi: 10.1016/j.healun.2008.10.012. Epub 2008 Dec 10.

Abstract

Background: The control of warm ischemia-reperfusion injury is crucial in managing donors after cardiac death for lung transplantation. We focused on transalveolar administration as a drug-delivery route for such donors. Milrinone is a phosphodiesterase 3 inhibitor that inhibits the breakdown of cyclic adenosine monophosphate and selectively relaxes smooth muscle. We hypothesized that nebulized milrinone would mitigate warm ischemia-reperfusion injury of lung.

Methods: This study was conducted with an isolated rat lung perfusion model. Lungs were excised, exposed to 55-minute ischemia at 37 degrees C, and reperfused for 60 minutes. During ischemia, nebulized milrinone (n = 6) or saline (n = 6) was inhaled. Lungs were continuously perfused without ischemia as a sham group (n = 6). Airway resistance, pulmonary vascular resistance, pulmonary compliance, weight gain and blood gas were measured. Adenine nucleotide levels and apoptosis were investigated in the reperfused lungs.

Results: Milrinone nebulization decreased post-ischemic pulmonary vascular resistance (0.98 +/- 0.05 and 1.74 +/- 0.17 cm H(2)O/ml.min at 60 minutes of reperfusion in the milrinone and control groups, respectively [p < 0.01]). It did not alter cyclic adenosine monophosphate levels, but it did elevate adenosine triphosphate levels (9.87 +/- 0.38 and 6.91 +/- 0.45 in the milrinone and control groups, respectively [p < 0.01]) and suppressed apoptosis (3.83 +/- 0.91 and 46.17 +/- 3.39 of mean apoptotic cell numbers in the milrinone and control groups, respectively [p < 0.01]).

Conclusions: Milrinone nebulization decreased post-ischemic pulmonary vascular resistance, elevated adenosine triphosphate levels, and suppressed apoptosis. Nebulized milrinone has some protective effects against warm ischemia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aerosols
  • Animals
  • DNA Nucleotidylexotransferase / metabolism
  • In Situ Nick-End Labeling
  • Lung / drug effects
  • Lung / physiology
  • Lung Transplantation / adverse effects
  • Lung Transplantation / physiology*
  • Male
  • Milrinone / administration & dosage
  • Milrinone / therapeutic use*
  • Models, Animal
  • Nebulizers and Vaporizers
  • Phosphodiesterase 3 Inhibitors*
  • Phosphodiesterase Inhibitors / administration & dosage
  • Phosphodiesterase Inhibitors / therapeutic use*
  • Postoperative Complications / prevention & control*
  • Rats
  • Reperfusion Injury / prevention & control*
  • Vascular Resistance / drug effects*

Substances

  • Aerosols
  • Phosphodiesterase 3 Inhibitors
  • Phosphodiesterase Inhibitors
  • DNA Nucleotidylexotransferase
  • Milrinone