The synthesis and in vivo evaluation of 2',2'-difluoro KRN7000

ChemMedChem. 2009 Mar;4(3):329-34. doi: 10.1002/cmdc.200800348.

Abstract

The synthesis of 2',2'-difluoro KRN7000 is described. In vivo evaluation demonstrates that this fluorinated glycolipid induces CD1d-dependent TCR activation of NKT cells, with a bias towards Th2 cytokine production.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigens, CD1 / immunology*
  • Cytokines / blood
  • Cytokines / immunology
  • Galactosylceramides / chemical synthesis*
  • Galactosylceramides / pharmacology*
  • Lymphocyte Activation / drug effects*
  • Mice
  • Mice, Inbred C57BL
  • Natural Killer T-Cells
  • Receptors, Natural Killer Cell / immunology

Substances

  • 2',2'-difluoro KRN7000
  • Antigens, CD1
  • Cytokines
  • Galactosylceramides
  • Receptors, Natural Killer Cell