Lipid A and related compounds. XXVI. Syntheses of biologically active penta-O-acetyl-N-glycoloylneuraminyl- and penta-O-acetyl-3-deoxy-D-galacto-2- nonulopyranosonic acid-(alpha 2----6)-D-glucosamine-4-phosphate analogs of lipid A

Chem Pharm Bull (Tokyo). 1991 May;39(5):1305-9. doi: 10.1248/cpb.39.1305.

Abstract

The syntheses of novel penta-O-acetyl-N-glycoloylneuraminyl- and penta-O-acetyl-3-deoxy-D-glycero-D-galacto-2-nonulopyranosonic acid-(alpha 2----6)-D-glucosamine-4-phosphate analogues of lipid A containing sialic acid in place of 3-deoxy-D-manno-2-octulosonic acid are described. Preliminary examination of the biological activity revealed that two synthetic disaccharides showed mitogenic activities and weak antitumor activities.

MeSH terms

  • Antineoplastic Agents / chemical synthesis
  • Antineoplastic Agents / pharmacology
  • Lipid A / analogs & derivatives*
  • Lipid A / chemical synthesis
  • Lipid A / pharmacology
  • Mitogens / chemical synthesis*
  • Mitogens / pharmacology

Substances

  • Antineoplastic Agents
  • Lipid A
  • Mitogens