Engineering heme binding sites in monomeric rop

J Biol Inorg Chem. 2009 May;14(4):497-505. doi: 10.1007/s00775-009-0465-0. Epub 2009 Jan 17.

Abstract

Heme ligands were introduced in the hydrophobic core of an engineered monomeric ColE1 repressor of primer (rop-S55) in two different layers of the heptad repeat. Mutants rop-L63M/F121H (layer 1) and rop-L56H/L113H (layer 3) were found to bind heme with a K (D) of 1.1 +/- 0.2 and 0.47 +/- 0.07 microM, respectively. The unfolding of heme-bound and heme-free mutants, in the presence of guanidinium hydrochloride, was monitored by both circular dichroism and fluorescence spectroscopy. For the heme-bound rop mutants, the total free energy change was 0.5 kcal/mol higher in the layer 3 mutant compared with that in the layer1 mutant. Heme binding also stabilized these mutants by increasing the [DGobsH2O] by 1.4 and 1.8 kcal/mol in rop-L63M/F121H and rop-L56H/L113H, respectively. The reduction potentials measured by spectroelectrochemical titrations were calculated to be -154 +/- 2 mV for rop-56H/113H and -87.5 +/- 1.2 mV for rop-L63M/F121H. The mutant designed to bind heme in a more buried environment (layer 3) showed tighter heme binding, a higher stability, and a different reduction potential compared with the mutant designed to bind heme in layer 1.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bacterial Proteins / chemistry*
  • Bacterial Proteins / genetics*
  • Bacterial Proteins / metabolism
  • Binding Sites
  • Electrochemistry
  • Heme / chemistry
  • Heme / metabolism*
  • Protein Binding
  • Protein Denaturation
  • Protein Engineering*
  • Protein Structure, Secondary
  • RNA-Binding Proteins / chemistry*
  • RNA-Binding Proteins / genetics*
  • RNA-Binding Proteins / metabolism
  • Thermodynamics

Substances

  • Bacterial Proteins
  • RNA-Binding Proteins
  • Rop protein, ColE1 plasmid
  • Heme