Efficient, regioselective palladium-catalyzed tandem Heck-isomerization reaction of aryl bromides and non-allylic benzyl alcohols

Org Lett. 2009 Mar 5;11(5):1183-5. doi: 10.1021/ol900036y.

Abstract

An efficient and mild method to couple aryl bromides and activated non-allylic alcohols in a Heck reaction with tandem isomerization to selectively afford high yields of 1,5-diarylalkan-1-ones has been developed. Mechanistic insight was gained through NMR studies of products derived from deuterium-labeled intermediates.

MeSH terms

  • Benzyl Alcohols / chemistry*
  • Bromides / chemistry*
  • Catalysis
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Palladium / chemistry*
  • Stereoisomerism

Substances

  • Benzyl Alcohols
  • Bromides
  • Palladium