Eslicarbazepine acetate: a new option for the treatment of focal epilepsy

Expert Opin Investig Drugs. 2009 Feb;18(2):221-9. doi: 10.1517/13543780802635107.

Abstract

Background: Epilepsy is a neurological condition with an increased probability of seizure occurrence through time. Although many anti-epileptic drugs (AEDs) exist, they fail to treat seizures in 30% of patients with epilepsy. For these patients, new AEDs potentially more efficacious and safe are developed.

Objective: To evaluate the effectiveness of eslicarbazepine acetate (ESL) in the treatment of patients with refractory epilepsy.

Methods: A review of the literature was carried out using PubMed central. A direct contact with the drug manufacturer and developer was made.

Results/conclusion: ESL is an AED that acts by inhibiting voltage-gated sodium channels. It has proved efficacious in the treatment of patients with refractory focal-onset epilepsy with a good safety profile. Evaluation of its use for treating other epileptic syndromes and its role as an initial treatment option for patients with epilepsy is warranted.

Publication types

  • Review

MeSH terms

  • Animals
  • Anticonvulsants / adverse effects
  • Anticonvulsants / chemistry
  • Anticonvulsants / pharmacokinetics
  • Anticonvulsants / therapeutic use*
  • Clinical Trials, Phase II as Topic
  • Clinical Trials, Phase III as Topic
  • Dibenzazepines / adverse effects
  • Dibenzazepines / chemistry
  • Dibenzazepines / pharmacokinetics
  • Dibenzazepines / therapeutic use*
  • Epilepsies, Partial / drug therapy*
  • Humans
  • Treatment Outcome

Substances

  • Anticonvulsants
  • Dibenzazepines
  • eslicarbazepine acetate