Rectal mucosa damage in rabbits after subchronical application of suppository bases

Pharm Res. 1991 Jul;8(7):945-50. doi: 10.1023/a:1015828201697.

Abstract

The effect of suppository bases on rabbit rectal mucosa was investigated using six triglyceride bases, polyethylene glycol, and a triglyceride base combined with monoglycerides or fatty acids and methyl esters of those acids. Rectal irritation was evaluated and scored according to defined pathological features. "Pure" triglycerides and a triglyceride to which a nonionic surfactant was added caused severe mucosal damage with ulceration and inflammation. Hyperemia was characteristic for irritation by polyethylene glycol suppositories. Mucosal damage by a pure triglyceride combined with monoglycerides or fatty acids and methyl esters of those acids was similar but statistically less pronounced than with all other bases.

MeSH terms

  • Animals
  • Excipients / toxicity*
  • Intestinal Mucosa / pathology*
  • Irritants
  • Male
  • Polyethylene Glycols
  • Rabbits
  • Rectal Diseases / chemically induced
  • Rectal Diseases / pathology*
  • Suppositories*
  • Triglycerides / toxicity

Substances

  • Excipients
  • Irritants
  • Suppositories
  • Triglycerides
  • Polyethylene Glycols