CD40 and B-cell receptor signalling induce MAPK family members that can either induce or repress Bcl-6 expression

Mol Immunol. 2009 May;46(8-9):1727-35. doi: 10.1016/j.molimm.2009.02.003. Epub 2009 Mar 6.

Abstract

Bcl-6 is essential for germinal centre development and normal antibody responses, and has major roles in controlling B-cell proliferation and differentiation. Bcl-6 expression is tightly controlled, but neither the nature of all the regulatory signals nor their interactions are known. Bcl-6 expression is induced in Bcr-Abl expressing lymphoid cell lines by the tyrosine kinase inhibitor, imatinib. We show that p38 MAPK mediates induction of Bcl-6 following inhibition of Bcr-Abl by imatinib. Next we analyze p38 function in a germinal centre B-cell line, Ramos. p38 is phosphorylated under basal conditions, and studies with p38 inhibitors show that it induces Bcl-6 expression. Membrane bound CD40 ligand activates p38 but also other MAPK pathways that strongly repress Bcl-6 and the overall effect is reduction in Bcl-6 expression. Surprisingly soluble CD40 ligand induces Bcl-6 by activating p38 without activating the repressive pathways. Hence different types of CD40 signalling are associated with varying effects on Bcl-6 expression. Transcription reporter assays demonstrate p38 responsive sequences at about 4.5 kb from the transcription start site. Immunocytochemistry of tonsil sections show phosphorylated p38 in a minor population of germinal centre B-cells. We demonstrate for the first time that p38 induces Bcl-6 transcription, but increased protein expression occurs only when the strong pathways repressing Bcl-6 are not activated.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Anti-Idiotypic / pharmacology
  • Blast Crisis / genetics
  • Blast Crisis / metabolism
  • CD40 Antigens / physiology*
  • Cell Line, Tumor
  • Cells, Cultured
  • Enzyme Activation / drug effects
  • Extracellular Signal-Regulated MAP Kinases / metabolism*
  • Fusion Proteins, bcr-abl / genetics
  • Fusion Proteins, bcr-abl / metabolism
  • Gene Expression Regulation / drug effects
  • Humans
  • K562 Cells
  • Leukemia, Myelogenous, Chronic, BCR-ABL Positive / genetics
  • Leukemia, Myelogenous, Chronic, BCR-ABL Positive / pathology
  • Models, Biological
  • Palatine Tonsil / drug effects
  • Palatine Tonsil / metabolism
  • Palatine Tonsil / pathology
  • Phosphorylation / drug effects
  • Proto-Oncogene Proteins c-bcl-6 / genetics*
  • Proto-Oncogene Proteins c-bcl-6 / metabolism
  • Receptors, Antigen, B-Cell / physiology*
  • Signal Transduction / physiology

Substances

  • Antibodies, Anti-Idiotypic
  • CD40 Antigens
  • Proto-Oncogene Proteins c-bcl-6
  • Receptors, Antigen, B-Cell
  • anti-IgM
  • Fusion Proteins, bcr-abl
  • Extracellular Signal-Regulated MAP Kinases