A simple and efficient route for preparing 2,3,5,6-tetraaminopyridine hydrochloride salt

Molecules. 2009 Apr 27;14(5):1652-9. doi: 10.3390/molecules14051652.

Abstract

A simple and efficient route for preparing 2,3,5,6-tetraaminopyridine hydrochloride salt (TAP x 3HCl x H(2)O) was introduced in this paper. The title compound was synthesized, as usual, in two steps (nitration and hydrogenation) with a total yield of 90%. The use of an oleum and fuming nitric acid mixture in the nitration step improved the yield and purity of the intermediate product. A highly efficient hydrogenation using a H(2)/Pd/C/C(2)H(5)OH system was developed. The products were characterized by TG, IR, (1)H-NMR, (13)C-NMR, HPLC and elemental analysis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminopyridines / chemical synthesis*
  • Aminopyridines / chemistry
  • Hydrogenation
  • Molecular Structure
  • Nitric Acid / chemistry
  • Salts / chemical synthesis*
  • Salts / chemistry

Substances

  • Aminopyridines
  • Salts
  • Nitric Acid